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LDHA-IN-3
CAS No. 227010-33-5
LDHA-IN-3( —— )
Catalog No. M35158 CAS No. 227010-33-5
LDHA-IN-3 (1-(phenylseleno)-4-(trifluoromethyl) benzene) is a potent non-competitive lactate dehydrogenase (LDHA) inhibitor with an IC50 value of 145.2 nM.LDHA-IN-3 is a selenobenzene compound that can be used in cancer research.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 126 | In Stock |
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| 5MG | 116 | In Stock |
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| 10MG | 186 | In Stock |
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| 25MG | 392 | In Stock |
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| 50MG | 535 | In Stock |
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| 100MG | 731 | In Stock |
|
| 200MG | 1004 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameLDHA-IN-3
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NoteResearch use only, not for human use.
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Brief DescriptionLDHA-IN-3 (1-(phenylseleno)-4-(trifluoromethyl) benzene) is a potent non-competitive lactate dehydrogenase (LDHA) inhibitor with an IC50 value of 145.2 nM.LDHA-IN-3 is a selenobenzene compound that can be used in cancer research.
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DescriptionLDHA-IN-3, as a selenobenzene compound, is a potent, noncompetitive lactate dehydrogenase (LDHA) inhibitor (IC50=145.2 nM). LDHA-IN-3 can be used for the research of cancer.
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In VitroCell Viability Assay Cell Line:MCF-7 cells Concentration:0~500 μM Incubation Time:48 hours Result:Showed cytotoxic effect.
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In Vivo——
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Synonyms——
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PathwayMetabolic Enzyme/Protease
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TargetDehydrogenase
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RecptorDehydrogenase
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Research Area——
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Indication——
Chemical Information
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CAS Number227010-33-5
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Formula Weight301.17
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Molecular FormulaC13H9F3Se
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 100 mg/mL (332.04 mM; Ultrasonic )
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SMILES[Se](C1=CC=C(C(F)(F)F)C=C1)C2=CC=CC=C2
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Kim EY, et al. A Novel Lactate Dehydrogenase Inhibitor, 1-(Phenylseleno)-4-(Trifluoromethyl) Benzene, Suppresses Tumor Growth through Apoptotic Cell Death. Sci Rep. 2019;9(1):3969. Published 2019 Mar 8.
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