Glutaminase-IN-3

CAS No. 1439399-45-7

Glutaminase-IN-3( —— )

Catalog No. M34941 CAS No. 1439399-45-7

Glutaminase-IN-3 is a potent Glutaminase 1 inhibitor with potential antitumor activity and inhibits GLS1 for cancer research.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 67 In Stock
5MG 54 In Stock
10MG 77 In Stock
25MG 122 In Stock
50MG 176 In Stock
100MG 259 In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    Glutaminase-IN-3
  • Note
    Research use only, not for human use.
  • Brief Description
    Glutaminase-IN-3 is a potent Glutaminase 1 inhibitor with potential antitumor activity and inhibits GLS1 for cancer research.
  • Description
    Glutaminase-IN-3 (compound 657) is a potent glutaminase inhibitor with an IC50 of 0.24 μM for Glutaminase 1 (GLS1). Glutaminase-IN-3 is extracted from patent WO2014089048A1, compound 657.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    Glutaminase
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1439399-45-7
  • Formula Weight
    452.45
  • Molecular Formula
    C19H19F3N6O2S
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 50 mg/mL (110.51 mM; Ultrasonic )
  • SMILES
    FC(F)(F)Oc1cccc(CC(=O)N=c2ccc(CCCCc3n[nH]c(=N)s3)n[nH]2)c1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Mark K. Bennett, et al. Treatment of cancer with heterocyclic inhibitors of glutaminase. WO2014089048A1.
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