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Dalcotidine

CAS No. 120958-90-9

Dalcotidine( —— )

Catalog No. M34564 CAS No. 120958-90-9

Dalcotidine (KU 1257) is a novel histamine H2 receptor antagonist with histamine H9 receptor antagonistic activity and antisecretory effects.

Purity : >98% (HPLC)

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

Size	Price / USD	Stock	Quantity
1 mL x 10 mM in DMSO	143	In Stock
5MG	143	In Stock
10MG	212	In Stock
25MG	343	In Stock
50MG	486	In Stock
100MG	684	In Stock
200MG	923	In Stock
500MG	Get Quote	In Stock
1G	Get Quote	In Stock

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Biological Information

Product Name

Dalcotidine
Note

Research use only, not for human use.
Brief Description

Dalcotidine (KU 1257) is a novel histamine H2 receptor antagonist with histamine H9 receptor antagonistic activity and antisecretory effects.
Description

Dalcotidine (KU 1257) is a novel histamine H2 receptor antagonist with histamine H9 receptor antagonistic activity and antisecretory effects.The Ki value for binding to guinea pig cerebral cortex was 0.040 The KB value for antagonism of histamine-induced positive chronotropic responses in the right atrium of isolate guinea pigs was 0.041.Dalcotidine improves the quality of ulcer healing, and may contribute to a reduction in ulcer recurrence and relapse rates.
In Vitro

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In Vivo

——
Synonyms

——
Pathway

GPCR/G Protein
Target

Histamine Receptor
Recptor

Histamine Receptor
Research Area

——
Indication

——

Chemical Information

CAS Number

120958-90-9
Formula Weight

319.44
Molecular Formula

C18H29N3O2
Purity

>98% (HPLC)
Solubility

——
SMILES

C(C1=CC(OCCCNC(NCC)=O)=CC=C1)N2CCCCC2
Chemical Name

——

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

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