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Ticolubant

CAS No. 154413-61-3

Ticolubant( —— )

Catalog No. M34447 CAS No. 154413-61-3

Ticolubant is orally active leukotriene B4 antagonist with high affinity for the human neutrophil LTB4 receptor (Ki = 0.78 nM), blocks LTB4-induced Ca2+ migration with an IC50 of 6.6 ± 1.5 nM, and shows topical anti-inflammatory activity in a mouse model of skin inflammation.

Purity : >98% (HPLC)

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Size	Price / USD	Stock	Quantity
5MG	302	In Stock
10MG	437	In Stock
25MG	673	In Stock
50MG	918	In Stock
100MG	1256	In Stock
200MG	1702	In Stock
500MG	Get Quote	In Stock
1G	Get Quote	In Stock

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Biological Information

Product Name

Ticolubant
Note

Research use only, not for human use.
Brief Description

Ticolubant is orally active leukotriene B4 antagonist with high affinity for the human neutrophil LTB4 receptor (Ki = 0.78 nM), blocks LTB4-induced Ca2+ migration with an IC50 of 6.6 ± 1.5 nM, and shows topical anti-inflammatory activity in a mouse model of skin inflammation.
Description

Ticolubant is orally active leukotriene B4 antagonist with high affinity for the human neutrophil LTB4 receptor (Ki = 0.78 nM), blocks LTB4-induced Ca2+ migration with an IC50 of 6.6 ± 1.5 nM, and shows topical anti-inflammatory activity in a mouse model of skin inflammation.
In Vitro

——
In Vivo

——
Synonyms

——
Pathway

GPCR/G Protein
Target

Calcium Channel
Recptor

Calcium Channel | LTR
Research Area

——
Indication

——

Chemical Information

CAS Number

154413-61-3
Formula Weight

460.37
Molecular Formula

C23H19Cl2NO3S
Purity

>98% (HPLC)
Solubility

——
SMILES

C(=C/C(O)=O)\C1=C(OCCC2=CC=CC=C2)C=CC(CSC3=C(Cl)C=CC=C3Cl)=N1
Chemical Name

——

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

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