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GSK299115A
CAS No. 864082-35-9
GSK299115A( —— )
Catalog No. M34272 CAS No. 864082-35-9
GSK299115A (GSK-299115A) is a selective ROCK1 Inhibitor. GSK299115A exhibits IC50 of 8nM, 620nM, 560nM for ROCK1, RSK1, p70S6K, respectively.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 945 | In Stock |
|
| 5MG | 772 | In Stock |
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| 10MG | 1074 | In Stock |
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| 25MG | 1596 | In Stock |
|
| 50MG | 2102 | In Stock |
|
| 100MG | 2762 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameGSK299115A
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NoteResearch use only, not for human use.
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Brief DescriptionGSK299115A (GSK-299115A) is a selective ROCK1 Inhibitor. GSK299115A exhibits IC50 of 8nM, 620nM, 560nM for ROCK1, RSK1, p70S6K, respectively.
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DescriptionGSK299115A is a G Protein-coupled Receptor Kinase (GRK) and PKA inhibitor.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayOthers
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TargetGRK (GPCRK)
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RecptorGRK
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Research Area——
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Indication——
Chemical Information
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CAS Number864082-35-9
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Formula Weight415.27
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Molecular FormulaC20H16Cl2N4O2
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Purity>98% (HPLC)
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Solubility——
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SMILESC(NC=1C=C2C(=CC1)NN=C2)(=O)C=3C(CC(=O)NC3C)C4=CC(Cl)=C(Cl)C=C4
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Homan KT, et al. Identification and structure-function analysis of subfamily selective G protein-coupled receptor kinase inhibitors. ACS Chem Biol. 2015 Jan 16;10(1):310-9. ?
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