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Tiospirone
CAS No. 87691-91-6
Tiospirone( —— )
Catalog No. M34041 CAS No. 87691-91-6
Tiospirone (BMY 13859-1 free base) is a 5-HT2 receptor antagonist and dopamine blocker that inhibits D2, 5-HT1a, 5-HT7, and sigma receptors.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 201 | Get Quote |
|
| 5MG | 309 | Get Quote |
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| 10MG | 567 | Get Quote |
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| 25MG | 881 | Get Quote |
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| 50MG | 1187 | Get Quote |
|
| 100MG | 1557 | Get Quote |
|
| 500MG | Get Quote | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameTiospirone
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NoteResearch use only, not for human use.
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Brief DescriptionTiospirone (BMY 13859-1 free base) is a 5-HT2 receptor antagonist and dopamine blocker that inhibits D2, 5-HT1a, 5-HT7, and sigma receptors.
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DescriptionTiospirone is a 5-HT2 receptor antagonist with affinity for D2, 5-HT1a, and 5-HT7, and sigma receptors. Tiospirone decreases consumption of ethanol while increasing food intake of rats. Tiospirone can also reduce the reinforcing properties of Cocaine exhibited in the conditioned place preference paradigm.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayGPCR/G Protein
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TargetDopamine Receptor
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RecptorDopamine Receptor | 5-HT Receptor
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Research Area——
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Indication——
Chemical Information
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CAS Number87691-91-6
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Formula Weight440.6
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Molecular FormulaC24H32N4O2S
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Purity>98% (HPLC)
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Solubility——
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SMILESO=C1N(C(=O)CC2(C1)CCCC2)CCCCN3CCN(C4=NSC=5C=CC=CC54)CC3
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Arolfo MP, et, al. Effects of amperozide and tiospirone, atypical antipsychotic 5-HT2 drugs, on food-reinforced behavior in rats. Physiol Behav. 1999 Dec;68(1-2):93-8.?
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