MK 1903

CAS No. 1268882-43-4

MK 1903( —— )

Catalog No. M33887 CAS No. 1268882-43-4

MK 1903 is a potent and selective complete agonist for the hydroxy-carboxylic acid receptor 2 (HCA2). HCA2 is also known as G protein-coupled receptor 109A(GPR109A).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 64 In Stock
5MG 93 In Stock
10MG 140 In Stock
25MG 242 In Stock
50MG 339 In Stock
100MG 466 In Stock
500MG Get Quote In Stock
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Biological Information

  • Product Name
    MK 1903
  • Note
    Research use only, not for human use.
  • Brief Description
    MK 1903 is a potent and selective complete agonist for the hydroxy-carboxylic acid receptor 2 (HCA2). HCA2 is also known as G protein-coupled receptor 109A(GPR109A).
  • Description
    MK-1903 is a potent and selective hydroxycarboxylic acid receptor 2 (HCA2, GPR109A) full agonist.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Cell Cycle/DNA Damage
  • Target
    GPR
  • Recptor
    GPR
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1268882-43-4
  • Formula Weight
    164.16
  • Molecular Formula
    C8H8N2O2
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 125 mg/mL (761.45 mM; Ultrasonic )
  • SMILES
    [H][C@]12C[C@@]1([H])c1[nH]nc(C(O)=O)c1C2
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Boatman PD, et al. (1aR,5aR)1a,3,5,5a-Tetrahydro-1H-2,3-diaza-cyclopropa[a]pentalene-4-carboxylic acid (MK-1903): a potent GPR109a agonist that lowers free fatty acids in humans. J Med Chem. 2012 Apr 26;55(8):3644-66.?
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