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ICI 204,448
CAS No. 121264-04-8
ICI 204,448( —— )
Catalog No. M33869 CAS No. 121264-04-8
ICI 204,448 is a potent κ-opioid agonist with potential analgesic activity for the study of neurological diseases.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 75 | In Stock |
|
| 10MG | 119 | In Stock |
|
| 25MG | 198 | In Stock |
|
| 50MG | 295 | In Stock |
|
| 100MG | Get Quote | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameICI 204,448
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NoteResearch use only, not for human use.
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Brief DescriptionICI 204,448 is a potent κ-opioid agonist with potential analgesic activity for the study of neurological diseases.
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DescriptionICI-204448 is a κ-opioid agonist with limited access to the CNS, ICI-204448 can displace the binding of the kappa-opioid ligand 3H-bremazocine from guinea pig cerebellum membranes.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayEndocrinology/Hormones
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TargetOpioid Receptor
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RecptorOpioid Receptor
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Research Area——
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Indication——
Chemical Information
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CAS Number121264-04-8
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Formula Weight501.83
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Molecular FormulaC23H27Cl3N2O4
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 125 mg/mL (249.09 mM; Ultrasonic )
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SMILESCl.O=C(O)COC1=CC=CC(=C1)C(N(C(=O)CC2=CC=C(Cl)C(Cl)=C2)C)CN3CCCC3
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. J S Shaw, et, al. ICI 204448: a kappa-opioid agonist with limited access to the CNS. Br J Pharmacol. 1989, 96, 4.?
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