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ICI 199,441 hydrochloride
CAS No. 115199-84-3
ICI 199,441 hydrochloride( —— )
Catalog No. M33868 CAS No. 115199-84-3
ICI 199,441 hydrochloride is a potent, selective agonist of κ-opioid receptor.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 53 | In Stock |
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| 2MG | 28 | In Stock |
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| 5MG | 44 | In Stock |
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| 10MG | 69 | In Stock |
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| 25MG | 141 | In Stock |
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| 50MG | 221 | In Stock |
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| 100MG | 325 | In Stock |
|
| 200MG | 456 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameICI 199,441 hydrochloride
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NoteResearch use only, not for human use.
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Brief DescriptionICI 199,441 hydrochloride is a potent, selective agonist of κ-opioid receptor.
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DescriptionICI 199441 is a potent and selective κ-opioid receptor agonist. ICI 199441 can improve heart resistance to ischemia/reperfusion.
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In Vitro——
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In VivoICI 199441 (Wistar rats, 0.1 mg/kg, IV, once) administered 15 min before ischemia produces a potent antiarrhythmic effect.
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Synonyms——
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PathwayEndocrinology/Hormones
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TargetOpioid Receptor
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RecptorOpioid Receptor
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Research Area——
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Indication——
Chemical Information
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CAS Number115199-84-3
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Formula Weight427.8
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Molecular FormulaC21H25Cl3N2O
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 250 mg/mL (584.39 mM; Ultrasonic )
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SMILESCl.CN([C@H](CN1CCCC1)c1ccccc1)C(=O)Cc1ccc(Cl)c(Cl)c1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Tsibulnikov SY, et al. Prospects of Using of κ-Opioid Receptor Agonists U-50,488 and ICI 199,441 for Improving Heart Resistance to Ischemia/Reperfusion. Bull Exp Biol Med. 2015;159(6):718-721.?
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