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Tenidap
CAS No. 120210-48-2
Tenidap( —— )
Catalog No. M33516 CAS No. 120210-48-2
Tenidap (CP-66248) is a selective COX-1 and SLC26A3 inhibitor with anti-inflammatory, analgesic, and anti-rheumatic activities.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 61 | In Stock |
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| 5MG | 55 | In Stock |
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| 10MG | 93 | In Stock |
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| 25MG | 201 | In Stock |
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| 50MG | 328 | In Stock |
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| 100MG | 573 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameTenidap
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NoteResearch use only, not for human use.
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Brief DescriptionTenidap (CP-66248) is a selective COX-1 and SLC26A3 inhibitor with anti-inflammatory, analgesic, and anti-rheumatic activities.
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DescriptionTenidap, a non-steroidal anti-inflammatory drug, is a selective COX-1 inhibitor, with IC50 values of 0.03 μM and 1.2 μM for COX-1 and COX-2, respectively. Tenidap has anti-inflammatory and antirheumatic properties. Tenidap is also a specific SLC26A3 inhibitor.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayChromatin/Epigenetic
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TargetCOX
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RecptorCOX | DNA/RNA Synthesis
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Research Area——
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Indication——
Chemical Information
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CAS Number120210-48-2
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Formula Weight320.75
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Molecular FormulaC14H9ClN2O3S
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 25 mg/mL (77.94 mM; Ultrasonic )
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SMILESNC(=O)N1C(=O)\C(=C(/O)c2cccs2)c2cc(Cl)ccc12
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Kirchner T, et al. Evaluation of the antiinflammatory activity of a dual cyclooxygenase-2 selective/5-lipoxygenase inhibitor, RWJ 63556, in a canine model of inflammation. J Pharmacol Exp Ther. 1997 Aug;282(2):1094-101.?
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