ZK-90055 hydrochloride

Research use only, not for human use.

ZK-90055 hydrochloride, a β2 adrenergic receptor agonist, is employed in the study of asthma.

ZK-90055 hydrochloride is a β2 adrenergic receptor agonist.

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Contrasting a pro-drug, a soft-drug is active per se when given locally but is rapidly inactivated when it reaches the general circulation. Thus, a long duration of action at a minimum of systemic side effects may be achieved after inhalation of a h2-agonist designed in this way. One such example is ZK-90055, an indol derivative with a hydrolysable ester bond on the ring system. The development of ZK-90055 is stopped before clinical trials are commenced.

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GPCR/G Protein

Adrenergic Receptor

Adrenergic Receptor

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84638-81-3

342.82

C16H23ClN2O4

>98% (HPLC)

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Cl.O=C(OC)C1=CC=2C(N1)=C(O)C=CC2C(O)CNC(C)(C)C

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(-20℃)

With Ice Pack

≥ 2 years