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RAS GTPase inhibitor 1
CAS No. 2252242-32-1
RAS GTPase inhibitor 1( —— )
Catalog No. M33100 CAS No. 2252242-32-1
RAS GTPase inhibitor 1 is a RAS GTPase inhibitor with potential antitumor activity.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 848 | Get Quote |
|
| 10MG | 1159 | Get Quote |
|
| 100MG | Get Quote | Get Quote |
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| 200MG | Get Quote | Get Quote |
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| 500MG | Get Quote | Get Quote |
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| 1G | Get Quote | Get Quote |
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Biological Information
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Product NameRAS GTPase inhibitor 1
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NoteResearch use only, not for human use.
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Brief DescriptionRAS GTPase inhibitor 1 is a RAS GTPase inhibitor with potential antitumor activity.
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DescriptionRAS GTPase inhibitor 1 (example 51) is a RAS GTPase inhibitor with anti-tumor activity, extracted from patent WO2018212774A1. RAS GTPase inhibitor 1 (example 51) exhibits an EC50 less than 1 μM for at least one nucleotide exchange and an IC50 less than 1 μM in H727 cells.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayMAPK/ERK Signaling
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TargetRaf
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RecptorRaf
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Research Area——
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Indication——
Chemical Information
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CAS Number2252242-32-1
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Formula Weight565.99
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Molecular FormulaC27H28ClF4N5O2
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Purity>98% (HPLC)
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Solubility——
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SMILESC(C(O)=O)(F)(F)F.N([C@H](CC)C1CC1)C=2C3=C(C(=CC=C3)C=4CCNCC4)N=C(NC5=CC(Cl)=C(F)C=C5)N2
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. WATERSON, Alex G, et al. QUINAZOLINE COMPOUNDS AS MODULATORS OF RAS SIGNALING. Patent. WO2018212774A1.
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