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ORM-10103
CAS No. 488847-28-5
ORM-10103( —— )
Catalog No. M33047 CAS No. 488847-28-5
ORM-10103 is a novel potent and selective inhibitor of the Na+/Ca2+ exchanger (NCX).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 132 | Get Quote |
|
| 10MG | 217 | Get Quote |
|
| 25MG | 447 | Get Quote |
|
| 50MG | 719 | Get Quote |
|
| 100MG | 954 | Get Quote |
|
| 500MG | 1917 | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameORM-10103
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NoteResearch use only, not for human use.
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Brief DescriptionORM-10103 is a novel potent and selective inhibitor of the Na+/Ca2+ exchanger (NCX).
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DescriptionORM-10103 is a specific inhibitor of the Na+/Ca2+ exchanger (NCX), which decreases the NCX current with estimated IC50s of 55 and 67 nM at -80 and at 20 mV, respectively.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayGPCR/G Protein
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TargetCalcium Channel
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RecptorCalcium Channel
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Research Area——
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Indication——
Chemical Information
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CAS Number488847-28-5
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Formula Weight348.35
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Molecular FormulaC20H16N2O4
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 250 mg/mL (717.67 mM; Ultrasonic )
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SMILES[O-][N+](=O)c1ccc(Oc2ccc3OC(CCc3c2)c2ccccc2)nc1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Jost N, et al. ORM-10103, a novel specific inhibitor of the Na+/Ca2+ exchanger, decreases early and delayed afterdepolarizations in the canine heart. Br J Pharmacol. 2013 Oct;170(4):768-78.?
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