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BIBF 1202
CAS No. 894783-71-2
BIBF 1202( —— )
Catalog No. M29632 CAS No. 894783-71-2
BIBF 1202 is a VEGFR2 kinase inhibitor (IC50 = 62 nM).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 61 | In Stock |
|
| 25MG | 179 | In Stock |
|
| 50MG | 259 | In Stock |
|
| 100MG | 379 | In Stock |
|
| 200MG | 537 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameBIBF 1202
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NoteResearch use only, not for human use.
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Brief DescriptionBIBF 1202 is a VEGFR2 kinase inhibitor (IC50 = 62 nM).
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DescriptionBIBF 1202 is a VEGFR2 kinase inhibitor (IC50 = 62 nM).(In Vitro):BIBF 1202 is produced in the main metabolic pathway of BIBF 1120 by the cleavage of methyl esters. Then, the free carboxyl group of BIBF 1202 is glucuronidated to 1-O-acyl glucuronide .
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In VitroThe major metabolic pathway for BIBF 1120 is methyl ester cleavage to BIBF 1202. Subsequently, the free carboxyl group of BIBF 1202 is glucuronidated to 1-O-acylglucuronide.
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In Vivo——
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Synonyms——
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PathwayAngiogenesis
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TargetVEGFR
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RecptorVEGFR
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Research Area——
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Indication——
Chemical Information
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CAS Number894783-71-2
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Formula Weight525.609
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Molecular FormulaC30H31N5O4
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : ≥ 45 mg/mL (85.62 mM)
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SMILESCN(C(=O)CN1CCN(C)CC1)c1ccc(N\C(=C2/C(=O)Nc3cc(ccc23)C(O)=O)c2ccccc2)cc1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
molnova catalog
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