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Histrelin acetate
CAS No. 220810-26-4
Histrelin acetate( Histrelin acetate(76712-82-8 free base) )
Catalog No. M29587 CAS No. 220810-26-4
Histrelin acetate is a nonapeptide analog of gonadotropin-releasing hormone (GnRH) with added potency. It acts on particular cells of the pituitary gland called gonadotropes when present in the bloodstream. Histrelin stimulates these cells to release luteinizing hormone and follicle-stimulating hormone. Thus it is considered a gonadotropin-releasing hormone agonist or GnRH agonist.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 169 | In Stock |
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| 10MG | 275 | In Stock |
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| 25MG | 465 | In Stock |
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| 50MG | 638 | In Stock |
|
| 100MG | 901 | In Stock |
|
| 200MG | Get Quote | In Stock |
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| 500MG | Get Quote | In Stock |
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| 1G | Get Quote | In Stock |
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Biological Information
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Product NameHistrelin acetate
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NoteResearch use only, not for human use.
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Brief DescriptionHistrelin acetate is a nonapeptide analog of gonadotropin-releasing hormone (GnRH) with added potency. It acts on particular cells of the pituitary gland called gonadotropes when present in the bloodstream. Histrelin stimulates these cells to release luteinizing hormone and follicle-stimulating hormone. Thus it is considered a gonadotropin-releasing hormone agonist or GnRH agonist.
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DescriptionHistrelin acetate is a nonapeptide analog of gonadotropin-releasing hormone (GnRH) with added potency. It acts on particular cells of the pituitary gland called gonadotropes when present in the bloodstream. Histrelin stimulates these cells to release luteinizing hormone and follicle-stimulating hormone. Thus it is considered a gonadotropin-releasing hormone agonist or GnRH agonist.
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In Vitro——
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In Vivo——
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SynonymsHistrelin acetate(76712-82-8 free base)
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PathwayOthers
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TargetOther Targets
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Recptor——
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Research Area——
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Indication——
Chemical Information
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CAS Number220810-26-4
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Formula Weight1383.55
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Molecular FormulaC68H90N18O14
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Purity>98% (HPLC)
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SolubilityIn Vitro:?H2O : 100 mg/mL
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SMILESCCNC([C@@H]1CCCN1C([C@H](CCCNC(N)=N)NC([C@H](CC(C)C)NC([C@@H](CC2=CN(C=N2)CC3=CC=CC=C3)NC([C@H](CC4=CC=C(C=C4)O)NC([C@H](CO)NC([C@H](CC5=CNC6=CC=CC=C65)NC([C@H](CC7=CNC=N7)NC([C@@H]8CCC(N8)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O.CC(O)=O
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
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Suc-Leu-Leu-Val-Tyr-...
Suc-Leu-Leu-Val-Tyr-AMC is a fluorescent substrate for the 20S proteasome, other chymotrypsin-like proteases.
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Head activator
Head activator neuropeptide is a mitogen for mammalian cell lines of neuronal or neuroendocrine origin. Head activator neuropeptide signals by binding GPR37 and stimulates cells to enter mitosis.
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CALP1
Cell-permeable calmodulin (CaM) agonist that binds to the EF-hand/Ca2+-binding site; produces CaM-dependent activation of phosphodiesterase. Also binds to cytoplasmic sites on other Ca2+ channels, including NMDA and HIV-1 gp120-activated channels, inhibiting Ca2+-mediated cytotoxicity and apoptosis (IC50 = 52 μM). Shown to protect pancreatic acinar cells from gossypol induced necrosis. Inhibits VLA-5-mediated adhesion of mast cells to fibronectin in vitro and attenuates inflammatory cell influx in guinea pig lung in vivo.
