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Ro 5212773
CAS No. 1110781-88-8
Ro 5212773( EPPTB | Epptb | Ro 5212773 )
Catalog No. M28628 CAS No. 1110781-88-8
EPPTB is a selective TAAR1 antagonist.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 75 | In Stock |
|
| 5MG | 68 | In Stock |
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| 10MG | 122 | In Stock |
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| 25MG | 271 | In Stock |
|
| 50MG | 530 | In Stock |
|
| 100MG | 760 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameRo 5212773
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NoteResearch use only, not for human use.
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Brief DescriptionEPPTB is a selective TAAR1 antagonist.
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DescriptionEPPTB is a selective TAAR1 antagonist.(In Vivo):EPPTB prevents the reduction of the firing frequency of DA neurons induced by p-tyramine (p-tyr), a nonselective TAAR1 agonist. the EPPTB effects were absent in Taar1 knockout mice, ruling out off-target effects.
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In Vitro——
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In Vivo——
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SynonymsEPPTB | Epptb | Ro 5212773
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PathwayOthers
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TargetOther Targets
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RecptorEGFR
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Research Area——
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Indication——
Chemical Information
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CAS Number1110781-88-8
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Formula Weight378.39
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Molecular FormulaC20H21F3N2O2
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 100 mg/mL (264.28 mM)
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SMILESCCOc1cccc(NC(c(cc2)cc(C(F)(F)F)c2N2CCCC2)=O)c1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.John Emmerson Campbell, et al. Inhibitors of mutant forms of egfr. Patent WO2021133809A1.
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