CCF0058981

CAS No. 2708934-53-4

CCF0058981( —— )

Catalog No. M28541 CAS No. 2708934-53-4

CCF0058981 is a SARS-CoV-2 inhibitor with low nanomolar biochemical inhibition and efficacy in cellular models comparable to that of Remdesivir.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 52 In Stock
5MG 88 In Stock
10MG 155 In Stock
25MG 324 In Stock
50MG 439 In Stock
100MG 551 In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    CCF0058981
  • Note
    Research use only, not for human use.
  • Brief Description
    CCF0058981 is a SARS-CoV-2 inhibitor with low nanomolar biochemical inhibition and efficacy in cellular models comparable to that of Remdesivir.
  • Description
    CCF0058981 is a SARS-CoV-2 inhibitor with low nanomolar biochemical inhibition and efficacy in cellular models comparable to that of Remdesivir.
  • In Vitro
    CCF0058981 (CCF981) has cytopathic effect (CPE) inhibition (EC50=497 nM) and plaque reduction (EC50=558 nM) in vitro viral replication. CCF0058981 has the 50% cytotoxic concentration (CC50) in the CPE antiviral assay of >50 μM. CCF0058981 has a T1/2 of 21.1 min, a CLlnt of 141 mL/min?kg in Human liver microsomes.
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    NF-κB|NOS|ROS
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    2708934-53-4
  • Formula Weight
    442.9
  • Molecular Formula
    C24H19ClN6O
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 25 mg/mL (56.45 mM)
  • SMILES
    O=C(N(C=1C=CC(=CC1)C2=CN=CN2)CC=3C=CC=C(Cl)C3)CN4N=NC=5C=CC=CC54
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.C Li, et al.Compounds from the bark of Illicium tsaii and their anti-inflammatory activity. Planta Medica. 2014 July; 80.
molnova catalog
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