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Tiazofurin
CAS No. 60084-10-8
Tiazofurin( NSC 286193 | Riboxamide )
Catalog No. M28325 CAS No. 60084-10-8
Tiazofurin is a synthetic nucleoside analogue with antineoplastic activity. Tiazofurin is anabolized intracellularly to tiazole-4-carboxamide adenine dinucleotide (TAD), a potent inhibitor of IMP dehydrogenase (IMPDH) .
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 70 | In Stock |
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| 5MG | 69 | In Stock |
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| 10MG | 117 | In Stock |
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| 25MG | 188 | In Stock |
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| 50MG | 276 | In Stock |
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| 100MG | Get Quote | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameTiazofurin
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NoteResearch use only, not for human use.
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Brief DescriptionTiazofurin is a synthetic nucleoside analogue with antineoplastic activity. Tiazofurin is anabolized intracellularly to tiazole-4-carboxamide adenine dinucleotide (TAD), a potent inhibitor of IMP dehydrogenase (IMPDH) .
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DescriptionTiazofurin is a synthetic nucleoside analogue with antineoplastic activity. Tiazofurin is anabolized intracellularly to tiazole-4-carboxamide adenine dinucleotide (TAD), a potent inhibitor of IMP dehydrogenase (IMPDH) .
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In Vitro——
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In Vivo——
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SynonymsNSC 286193 | Riboxamide
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PathwayMetabolic Enzyme/Protease
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TargetDehydrogenase
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RecptorAntifungal
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Research Area——
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Indication——
Chemical Information
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CAS Number60084-10-8
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Formula Weight260.26
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Molecular FormulaC9H12N2O5S
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Purity>98% (HPLC)
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Solubility——
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SMILESNC(=O)c1csc(n1)[C@@H]1O[C@H](CO)[C@@H](O)[C@H]1O
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Moraes DC, et al. β-lapachone and α-nor-lapachone modulate Candida albicans viability and virulence factors. J Mycol Med. 2018 Mar 26. pii: S1156-5233(17)30379-7.
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