Cart
sales@molnova.com
Home - Products - Membrane Transporter/Ion Channel - TRP/TRPV Channel - MK-2295

MK-2295

CAS No. 878811-00-8

MK-2295( MK2295 | MK 2295 )

Catalog No. M27996 CAS No. 878811-00-8

MK-2295 is a potent TRPV1 antagonist. MK-2295 can be used in studies about the treatment of chronic pain.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 149 In Stock
10MG 220 In Stock
25MG 337 In Stock
50MG 462 In Stock
100MG 619 In Stock
200MG 835 In Stock
500MG Get Quote In Stock
1G Get Quote In Stock
Get Quotation Bulk Inquiry Add to Cart

Biological Information

  • Product Name
    MK-2295
  • Note
    Research use only, not for human use.
  • Brief Description
    MK-2295 is a potent TRPV1 antagonist. MK-2295 can be used in studies about the treatment of chronic pain.
  • Description
    MK-2295 is a potent TRPV1 antagonist. MK-2295 can be used in studies about the treatment of chronic pain.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    MK2295 | MK 2295
  • Pathway
    Membrane Transporter/Ion Channel
  • Target
    TRP/TRPV Channel
  • Recptor
    JAK1
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    878811-00-8
  • Formula Weight
    490.583
  • Molecular Formula
    C27H31FN6O2
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    C[C@@H]1CCCN1c1nc(cc(n1)-c1ccc(F)cc1)N1CCN(C[C@H]1C)c1ncc(cc1C)C(O)=O
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Paul Smith, et al. Use of jak1 inhibitors for the treatment of cutaneous lupus erythematosus and lichen planus (lp). WO2021076124A1.
Calculator

Molecular Weight Calculator

Dilution Calculator

Molarity Calculator

molnova catalog
related products

  • Pyr6

    Pyr6 is a selective TRPC3 inhibitor with IC50 of 0.49 uM(Ca2+ influx inhibition in thapsigargin depleted native RBL-2H3 cells).Pyr6 is an inhibitor of Ca2+ entry, which displays higher potency to inhibit Ca2+ entry mediated by CRAC channel than by TRPC3.Pyr3 is selective inhibitor of TRPC3, inhibited Orai1- and TRPC3-mediated Ca(2+) entry and currents as well as mast cell activation with similar potency.?

  • TRPM8 antagonist 3

    TRPM8 antagonist 3 is a blocker of TRPM8 (IC50 = 11 nM).

  • RN-1665

    RN-1665 is a potent and selective TRPV4 receptor antagonist.

Sign In Join Free