ABT 102

CAS No. 808756-71-0

ABT 102( ABT-102 | ABT102 | CHEMBL398338 )

Catalog No. M27944 CAS No. 808756-71-0

ABT 102 is a selective antagonist of transient receptor potential vanilloid 1 (TRPV1) receptor.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 258 In Stock
5MG 249 In Stock
10MG 369 In Stock
25MG 562 In Stock
50MG 770 In Stock
100MG 1032 In Stock
200MG 1376 In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    ABT 102
  • Note
    Research use only, not for human use.
  • Brief Description
    ABT 102 is a selective antagonist of transient receptor potential vanilloid 1 (TRPV1) receptor.
  • Description
    ABT 102 is a selective antagonist of transient receptor potential vanilloid 1 (TRPV1) receptor.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ABT-102 | ABT102 | CHEMBL398338
  • Pathway
    Membrane Transporter/Ion Channel
  • Target
    TRP/TRPV Channel
  • Recptor
    ——
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    808756-71-0
  • Formula Weight
    348.44
  • Molecular Formula
    C21H24N4O
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    O=C(NC1=CC=CC2=C1C=NN2)N[C@@H]3CCC4=C3C=CC(C(C)(C)C)=C4
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Nishiguchi G, et al. Identification of Potent, Selective, and Orally Bioavailable Small-Molecule GSPT1/2 Degraders from a Focused Library of Cereblon Modulators. J Med Chem. 2021 Jun 10;64(11):7296-7311.
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