ABT 102
CAS No. 808756-71-0
ABT 102( ABT-102 | ABT102 | CHEMBL398338 )
Catalog No. M27944 CAS No. 808756-71-0
ABT 102 is a selective antagonist of transient receptor potential vanilloid 1 (TRPV1) receptor.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 258 | In Stock |
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| 5MG | 249 | In Stock |
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| 10MG | 369 | In Stock |
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| 25MG | 562 | In Stock |
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| 50MG | 770 | In Stock |
|
| 100MG | 1032 | In Stock |
|
| 200MG | 1376 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameABT 102
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NoteResearch use only, not for human use.
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Brief DescriptionABT 102 is a selective antagonist of transient receptor potential vanilloid 1 (TRPV1) receptor.
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DescriptionABT 102 is a selective antagonist of transient receptor potential vanilloid 1 (TRPV1) receptor.
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In Vitro——
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In Vivo——
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SynonymsABT-102 | ABT102 | CHEMBL398338
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PathwayMembrane Transporter/Ion Channel
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TargetTRP/TRPV Channel
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Recptor——
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Research Area——
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Indication——
Chemical Information
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CAS Number808756-71-0
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Formula Weight348.44
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Molecular FormulaC21H24N4O
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Purity>98% (HPLC)
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Solubility——
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SMILESO=C(NC1=CC=CC2=C1C=NN2)N[C@@H]3CCC4=C3C=CC(C(C)(C)C)=C4
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Nishiguchi G, et al. Identification of Potent, Selective, and Orally Bioavailable Small-Molecule GSPT1/2 Degraders from a Focused Library of Cereblon Modulators. J Med Chem. 2021 Jun 10;64(11):7296-7311.
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