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FEMA-4809
CAS No. 1374760-95-8
FEMA-4809( —— )
Catalog No. M34249 CAS No. 1374760-95-8
FEMA-4809, a highly potent TRPM8 receptor activator, TRPM8 is the ion channel responsible for the cool perception.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 77 | In Stock |
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| 5MG | 67 | In Stock |
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| 10MG | 112 | In Stock |
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| 25MG | 190 | In Stock |
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| 50MG | 263 | In Stock |
|
| 100MG | 375 | In Stock |
|
| 200MG | 514 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameFEMA-4809
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NoteResearch use only, not for human use.
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Brief DescriptionFEMA-4809, a highly potent TRPM8 receptor activator, TRPM8 is the ion channel responsible for the cool perception.
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DescriptionFEMA 4809 is a TRPM8 receptor agonist (EC50=0.2 nM) for use as a cooling agent. TRPM8 is the ion channel responsible for the cool perception.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayMembrane Transporter/Ion Channel
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TargetTRP/TRPV Channel
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RecptorTRP/TRPV Channel
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Research Area——
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Indication——
Chemical Information
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CAS Number1374760-95-8
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Formula Weight327.4
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Molecular FormulaC17H17N3O2S
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 250 mg/mL (763.59 mM; Ultrasonic )
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SMILESCc1ccc(OCC(=O)N(Cc2cccs2)c2cc[nH]n2)cc1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Alain Noncovich, et al. Discovery and development of a novel class of phenoxyacetyl amides as highly potent TRPM8 agonists for use as cooling agents. Bioorg Med Chem Lett. 2017 Aug 15;27(16):3931-3938.?
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