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PD 174265
CAS No. 216163-53-0
PD 174265( PD174265 | PD-174265 | N-{4-[(3-Bromophenyl)amino]quinazolin-6-Yl}propanamide )
Catalog No. M27910 CAS No. 216163-53-0
PD 174265 is an effective, selective and reversible inhibitor of epidermal growth factor receptor (EGFR) with an IC50 of 0.45 nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 36 | In Stock |
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| 5MG | 29 | In Stock |
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| 10MG | 36 | In Stock |
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| 25MG | 54 | In Stock |
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| 50MG | 74 | In Stock |
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| 100MG | 108 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NamePD 174265
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NoteResearch use only, not for human use.
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Brief DescriptionPD 174265 is an effective, selective and reversible inhibitor of epidermal growth factor receptor (EGFR) with an IC50 of 0.45 nM.
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DescriptionPD 174265 is an effective, selective and reversible inhibitor of epidermal growth factor receptor (EGFR) with an IC50 of 0.45 nM.
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In Vitro——
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In Vivo——
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SynonymsPD174265 | PD-174265 | N-{4-[(3-Bromophenyl)amino]quinazolin-6-Yl}propanamide
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PathwayAngiogenesis
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TargetEGFR
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RecptorInfluenza Virus
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Research Area——
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Indication——
Chemical Information
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CAS Number216163-53-0
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Formula Weight371.238
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Molecular FormulaC17H15BrN4O
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 125 mg/mL (336.72 mM)
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SMILESCCC(=O)Nc1ccc2ncnc(Nc3cccc(Br)c3)c2c1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Takizawa N, et al. Anti-influenza virus activity of a salcomine derivative mediated by inhibition of viral RNA synthesis. Arch Virol. 2018 Jun;163(6):1607-1614.
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