Tecastemizole

CAS No. 75970-99-9

Tecastemizole( Norastemizole | R 43512 | R-43512 | R43512 | T 1348 )

Catalog No. M27833 CAS No. 75970-99-9

Tecastemizole is a selective antagonist of H1 receptor and a major metabolite of astemizole with anti-inflammatory effects.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 134 In Stock
5MG 121 In Stock
10MG 178 In Stock
25MG 303 In Stock
50MG 428 In Stock
100MG 603 In Stock
200MG Get Quote In Stock
500MG 1200 In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    Tecastemizole
  • Note
    Research use only, not for human use.
  • Brief Description
    Tecastemizole is a selective antagonist of H1 receptor and a major metabolite of astemizole with anti-inflammatory effects.
  • Description
    Tecastemizole is a selective antagonist of H1 receptor and a major metabolite of astemizole with anti-inflammatory effects.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    Norastemizole | R 43512 | R-43512 | R43512 | T 1348
  • Pathway
    GPCR/G Protein
  • Target
    Histamine Receptor
  • Recptor
    ——
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    75970-99-9
  • Formula Weight
    324.403
  • Molecular Formula
    C19H21FN4
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 100 mg/mL (308.26 mM)
  • SMILES
    Fc1ccc(Cn2c(NC3CCNCC3)nc3ccccc23)cc1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Bernd R?dle, et al.Metabolic labeling of newly transcribed RNA for high resolution gene expression profiling of RNA synthesis, processing and decay in cell culture. J Vis Exp. 2013 Aug 8;(78):50195.
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