TCS 46b

CAS No. 302799-86-6

TCS 46b( —— )

Catalog No. M27726 CAS No. 302799-86-6

TCS 46b is a NR1A/NR2B NMDA receptor antagonist with oral activity.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 98 Get Quote
10MG 158 Get Quote
25MG 335 Get Quote
50MG 537 Get Quote
100MG 888 Get Quote
500MG 1782 Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    TCS 46b
  • Note
    Research use only, not for human use.
  • Brief Description
    TCS 46b is a NR1A/NR2B NMDA receptor antagonist with oral activity.
  • Description
    TCS 46b is a NR1A/NR2B NMDA receptor antagonist with oral activity.
  • In Vitro
    ——
  • In Vivo
    Animal Model:Sprague?Dawley rats, 6-hydroxydopamine-lesioned (6-OHDA) rat modelDosage:10 and 30 mg/kg Administration:PO or IP, once Result:Showed significant potentiation of the effects of L-DOPA in this model.
  • Synonyms
    ——
  • Pathway
    Membrane Transporter/Ion Channel
  • Target
    NMDAR
  • Recptor
    ——
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    302799-86-6
  • Formula Weight
    345.446
  • Molecular Formula
    C22H23N3O
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 100 mg/mL (289.49 mM)
  • SMILES
    O=c1[nH]c2ccc(cc2[nH]1)C#CCN1CCC(Cc2ccccc2)CC1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Fdez Galván I, et al. Solvent Effects on the Structure and Spectroscopy of the Emitting States of 1-Phenylpyrrole. J Chem Theory Comput. 2011 Jun 14;7(6):1850-7.
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