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Sonepiprazole

CAS No. 170858-33-0

Sonepiprazole( PNU-101387G | U-101387G )

Catalog No. M27715 CAS No. 170858-33-0

Sonepiprazole (PNU-101387G) is a selective D4 dopamine antagonist with Kis of 3.6, 10.1, 5147, and 7430 nM for rD4-Dopamine, hD4.2-Dopamine, rD2-Dopamine, and Histamine-H1 receptors, respectively.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 44 In Stock
5MG 35 In Stock
10MG 57 In Stock
25MG 126 In Stock
50MG 210 In Stock
100MG 303 In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G Get Quote In Stock
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Biological Information

  • Product Name
    Sonepiprazole
  • Note
    Research use only, not for human use.
  • Brief Description
    Sonepiprazole (PNU-101387G) is a selective D4 dopamine antagonist with Kis of 3.6, 10.1, 5147, and 7430 nM for rD4-Dopamine, hD4.2-Dopamine, rD2-Dopamine, and Histamine-H1 receptors, respectively.
  • Description
    Sonepiprazole (PNU-101387G) is a selective D4 dopamine antagonist with Kis of 3.6, 10.1, 5147, and 7430 nM for rD4-Dopamine, hD4.2-Dopamine, rD2-Dopamine, and Histamine-H1 receptors, respectively.
  • In Vitro
    Sonepiprazole exhibits highly specific binding to the D4 dopamine receptor with more than 100-fold selectivity for the D4 receptor over other receptors, including dopamine, serotonin, and adrenergic receptors.
  • In Vivo
    ——
  • Synonyms
    PNU-101387G | U-101387G
  • Pathway
    GPCR/G Protein
  • Target
    Dopamine Receptor
  • Recptor
    NOX1
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    170858-33-0
  • Formula Weight
    401.53
  • Molecular Formula
    C21H27N3O3S
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 125 mg/mL (311.32 mM)
  • SMILES
    NS(=O)(=O)c1ccc(cc1)N1CCN(CC[C@H]2OCCc3ccccc23)CC1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Brown SJ, et al. Probe Report for NOX1 Inhibitors. 2009 Apr 23 [updated 2010 Sep 2]. In: Probe Reports from the NIH Molecular Libraries Program [Internet]. Bethesda (MD): National Center for Biotechnology Information (US); 2010–.
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