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PSN 375963
CAS No. 388575-52-8
PSN 375963( PSN 375963 hydrochloride | PSN 375963 )
Catalog No. M27691 CAS No. 388575-52-8
PSN 375963 hydrochloride is a synthetic agonist of the endogenous ligand for GPR119.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 55 | In Stock |
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| 5MG | 36 | In Stock |
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| 10MG | 56 | In Stock |
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| 25MG | 112 | In Stock |
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| 50MG | 183 | In Stock |
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| 100MG | 300 | In Stock |
|
| 200MG | 428 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NamePSN 375963
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NoteResearch use only, not for human use.
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Brief DescriptionPSN 375963 hydrochloride is a synthetic agonist of the endogenous ligand for GPR119.
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DescriptionPSN 375963 hydrochloride is a synthetic agonist of the endogenous ligand for GPR119.(In Vitro):PSN 375963 is a potent GPR119 agonist with EC50s of 8.4 and 7.9 μM for human and mouse GPR119.(In Vivo):PSN 375963 suppressed food intake in rats and reduced body weight gain and white adipose tissue deposition upon subchronic oral administration to high-fat-fed rats.
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In VitroThe endogenous ligand OEA signals through GPR119 in a manner similar to glucagon-like peptide-1 (GLP-1) and its receptor with respect to insulin secretion, intracellular calcium and cAMP.
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In Vivo——
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SynonymsPSN 375963 hydrochloride | PSN 375963
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PathwayCell Cycle/DNA Damage
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TargetGPR
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RecptorNDM-1
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Research Area——
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Indication——
Chemical Information
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CAS Number388575-52-8
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Formula Weight321.85
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Molecular FormulaC17H24ClN3O
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 50 mg/mL (175.20 mM)
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SMILESCl.CCCC[C@H]1CC[C@@H](CC1)c1nc(no1)-c1ccncc1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Cui-Gai Bai, et al. Cysteine and Its Derivatives as New Delhi Metallo-beta-lactamase-1 Inhibitors. Current Enzyme Inhibition, 2015, 11, 46-57
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