CP94253 hydrochloride

CAS No. 845861-39-4

CP94253 hydrochloride( CP 94253 hydrochloride )

Catalog No. M27617 CAS No. 845861-39-4

CP94253 hydrochloride is a potent, selective and centrally active agonist of 5-HT1B receptor with Ki of 2 nM. The Kis are 89, 49, 860, and 1600 nM for 5-HT1A, 5-HT1D, 5-HT1C and 5-HT2 receptors, respectively.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 61 In Stock
5MG 61 In Stock
10MG 92 In Stock
25MG 217 In Stock
50MG 346 In Stock
100MG 555 In Stock
200MG 770 In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    CP94253 hydrochloride
  • Note
    Research use only, not for human use.
  • Brief Description
    CP94253 hydrochloride is a potent, selective and centrally active agonist of 5-HT1B receptor with Ki of 2 nM. The Kis are 89, 49, 860, and 1600 nM for 5-HT1A, 5-HT1D, 5-HT1C and 5-HT2 receptors, respectively.
  • Description
    CP94253 hydrochloride is a potent, selective and centrally active agonist of 5-HT1B receptor with Ki of 2 nM. The Kis are 89, 49, 860, and 1600 nM for 5-HT1A, 5-HT1D, 5-HT1C and 5-HT2 receptors, respectively.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    CP 94253 hydrochloride
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    panx1|Topo IV|Bacterial|DNA-gyrase
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    845861-39-4
  • Formula Weight
    293.8
  • Molecular Formula
    C15H20ClN3O
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 125 mg/mL (425.47 mM)
  • SMILES
    Cl.CCCOc1ccc2[nH]cc(C3=CCNCC3)c2n1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Poon IK, et al. Unexpected link between an antibiotic, pannexin channels and apoptosis. Nature. 2014 Mar 20;507(7492):329-34.
molnova catalog
related products
  • Allatostatin II

    Inhibitors of juvenile hormone synthesis in insects.

  • coreopsin

    Coreopsin is one of the main components from Coreopsis tinctoria Nutt. Flower(CTF). CTF has been used traditionally in China for treating hypertension and diabetes as well as reducing body weight and blood fat.

  • EPI 743

    EPI 743 (Vatiquinone) is an orally bioavailable para-benzoquinone for treatment of inherited mitochondrial diseases, an analogue of the antioxidant ubidecarenone.