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A 77636 hydrochloride
CAS No. 145307-34-2
A 77636 hydrochloride( A77636 hydrochloride )
Catalog No. M27461 CAS No. 145307-34-2
A-77636 hydrochloride is a potent, orally active, selective and long acting dopamine D1 receptor agonist (pKi=7.40; Ki=39.8 nM).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 217 | In Stock |
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| 10MG | 316 | In Stock |
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| 25MG | 533 | In Stock |
|
| 50MG | 734 | In Stock |
|
| 100MG | Get Quote | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameA 77636 hydrochloride
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NoteResearch use only, not for human use.
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Brief DescriptionA-77636 hydrochloride is a potent, orally active, selective and long acting dopamine D1 receptor agonist (pKi=7.40; Ki=39.8 nM).
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DescriptionA-77636 hydrochloride is a potent, orally active, selective and long acting dopamine D1 receptor agonist (pKi=7.40; Ki=39.8 nM). A-77636 hydrochloride shows antiparkinsonian activity. A-77636 hydrochloride is functionally inactive at dopamine D2 receptor.(In Vivo):A-77636 (0.1-1 mg/kg) exerts a suppressant effect on food intake in male hooded rat, due principally to a reduction in meal size and duration.
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In Vitro——
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In VivoAnimal Model:Male hooded ratDosage:0.1, 0.3 and 1.0 mg/kg Administration:S.c.Result:Exerted a suppressant effect on food intake, due principally to a reduction in meal size and duration.
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SynonymsA77636 hydrochloride
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PathwayGPCR/G Protein
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TargetDopamine Receptor
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RecptorFree radical scavengers|Platelet aggregation
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Research Area——
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Indication——
Chemical Information
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CAS Number145307-34-2
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Formula Weight365.89
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Molecular FormulaC20H28ClNO3
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Purity>98% (HPLC)
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Solubility——
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SMILESC(N)[C@@H]1O[C@H]([C@@]23CC4CC(C2)CC(C3)C4)CC=5C1=CC=C(O)C5O.Cl
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Zbidi H, et al. Olive tree wood phenolic compounds with human platelet antiaggregant properties. Blood Cells Mol Dis. 2009 May-Jun;42(3):279-85.
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