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Talinolol

CAS No. 57460-41-0

Talinolol( (±)-Talinolol )

Catalog No. M27440 CAS No. 57460-41-0

(±)-Talinolol is a selective β1 adrenoceptor antagonist well known for its cardioprotective and antihypertensive activity.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    Talinolol
  • Note
    Research use only, not for human use.
  • Brief Description
    (±)-Talinolol is a selective β1 adrenoceptor antagonist well known for its cardioprotective and antihypertensive activity.
  • Description
    (±)-Talinolol is a selective β1 adrenoceptor antagonist well known for its cardioprotective and antihypertensive activity.
  • In Vitro
    Human OATP1A2-, rat Oatp1a5-, and rat Mdr1a-mediated Talinolol transport can be inhibited by naringin, with IC50s of 343, 12.7, and 604 μM, respectively, in LLC-PK1 cell and Xenopus laevis oocyte systems.
  • In Vivo
    Talinolol (20 mg/kg; i.p.) plasma and liver AUC0-5 h are increased by Zosuquidar administration.Bioavailability of Talinolol can be enhanced by coadministration with grapefruit juice (GFJ) in rats.
  • Synonyms
    (±)-Talinolol
  • Pathway
    Angiogenesis
  • Target
    Adrenergic Receptor
  • Recptor
    ——
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    57460-41-0
  • Formula Weight
    363.502
  • Molecular Formula
    C20H33N3O3
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 100 mg/mL (275.11 mM)
  • SMILES
    CC(C)(C)NCC(O)COc1ccc(NC(=O)NC2CCCCC2)cc1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Asano T, Murayama T, Hirai Y, Shoji J. Comparative studies on the constituents of ophiopogonis tuber and its congeners. VIII. Studies on the glycosides of the subterranean part of Ophiopogon japonicus Ker-Gawler cv. Nanus. Chem Pharm Bull (Tokyo). 1993;41
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