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ML-290
CAS No. 1482500-76-4
ML-290( —— )
Catalog No. M26758 CAS No. 1482500-76-4
ML-290 is an effective relaxin/insulin-like family peptide receptor (RXFP1) agonist and activator of anti-fibrotic genes. It shows an EC50 of 94 nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 533 | Get Quote |
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| 100MG | Get Quote | Get Quote |
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| 200MG | Get Quote | Get Quote |
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| 500MG | Get Quote | Get Quote |
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| 1G | Get Quote | Get Quote |
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Biological Information
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Product NameML-290
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NoteResearch use only, not for human use.
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Brief DescriptionML-290 is an effective relaxin/insulin-like family peptide receptor (RXFP1) agonist and activator of anti-fibrotic genes. It shows an EC50 of 94 nM.
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DescriptionML-290 is an effective relaxin/insulin-like family peptide receptor (RXFP1) agonist and activator of anti-fibrotic genes. It shows an EC50 of 94 nM.(In Vitro):ML290 (5 μM; 24 and 72 h) displays anti-fibrotic, relaxin-like gene expression in activated human hepatic stellate cells.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayOthers
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TargetOther Targets
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RecptormTOR
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Research Area——
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Indication——
Chemical Information
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CAS Number1482500-76-4
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Formula Weight506.5
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Molecular FormulaC24H21F3N2O5S
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 125 mg/mL (246.80 mM)
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SMILESCC(C)Oc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(c1)S(=O)(=O)C(F)(F)F
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Park JH, et al. Human cardiac stem cells rejuvenated by modulating autophagy with MHY-1685 enhance the therapeutic potential for cardiac repair. Exp Mol Med. 2021 Sep;53(9):1423-1436.
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