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NSC232003
CAS No. 1905453-18-0
NSC232003( —— )
Catalog No. M26342 CAS No. 1905453-18-0
NSC232003 is a highly potent and cell-permeable inhibitor of UHRF1.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 201 | In Stock |
|
| 10MG | 314 | In Stock |
|
| 25MG | 602 | In Stock |
|
| 50MG | 842 | In Stock |
|
| 100MG | 1134 | In Stock |
|
| 500MG | 2268 | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameNSC232003
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NoteResearch use only, not for human use.
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Brief DescriptionNSC232003 is a highly potent and cell-permeable inhibitor of UHRF1.
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DescriptionNSC232003 is a highly potent and cell-permeable inhibitor of UHRF1.(In Vitro):NSC232003 is an effective DNA methylation inhibitor and indicate that this particular nucleotide scaffold could provide a versatile basis for the design of potent UHRF1 inhibitors.NSC232003, a uracil derivative freely available by the NCI/DTP repository, provides a versatile lead for developing highly potent and cell-permeable UHRF1 inhibitors that will enable dissection of DNA methylation inheritance.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayProteasome/Ubiquitin
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TargetE1
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RecptorDP8/9| DPP-4
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Research Area——
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Indication——
Chemical Information
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CAS Number1905453-18-0
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Formula Weight169.14
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Molecular FormulaC6H7N3O3
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Purity>98% (HPLC)
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SolubilityIn Vitro:?H2O : 2 mg/mL (11.82 mM)
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SMILESC\C(NO)=C1/C=NC(=O)NC1=O
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Ansorge S, et al. Novel aspects of cellular action of dipeptidyl peptidase IV/CD26. Biol Chem. 2011 Mar;392(3):153-68.
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