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NMDA-IN-1
CAS No. 700878-19-9
NMDA-IN-1( —— )
Catalog No. M26334 CAS No. 700878-19-9
NMDA-IN-1 is a potent and NR2B-selective antagonist of NMDA(NMDA Ki of 0.85 nM; NR2B Ca2+ influx IC50 is 9.7 nM).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 205 | Get Quote |
|
| 10MG | 357 | Get Quote |
|
| 25MG | 587 | Get Quote |
|
| 50MG | 822 | Get Quote |
|
| 100MG | 1107 | Get Quote |
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| 200MG | Get Quote | Get Quote |
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| 500MG | Get Quote | Get Quote |
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| 1G | Get Quote | Get Quote |
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Biological Information
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Product NameNMDA-IN-1
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NoteResearch use only, not for human use.
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Brief DescriptionNMDA-IN-1 is a potent and NR2B-selective antagonist of NMDA(NMDA Ki of 0.85 nM; NR2B Ca2+ influx IC50 is 9.7 nM).
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DescriptionNMDA-IN-1 is a potent and NR2B-selective antagonist of NMDA(NMDA Ki of 0.85 nM; NR2B Ca2+ influx IC50 is 9.7 nM).
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayMembrane Transporter/Ion Channel
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TargetNMDAR
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RecptorPEGs
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Research Area——
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Indication——
Chemical Information
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CAS Number700878-19-9
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Formula Weight375.87
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Molecular FormulaC20H23ClFN3O
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 12.5 mg/mL (33.26 mM)
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SMILESCl.Oc1ccc2nc(CN3CCC(Cc4ccccc4F)CC3)[nH]c2c1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.An S, et al. Small-molecule PROTACs: An emerging and promising approach for the development of targeted therapy drugs. EBioMedicine. 2018 Oct;36:553-562
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