Ziconotide Acetate (107452-89-1 free base)
CAS No. 914451-03-8
Ziconotide Acetate (107452-89-1 free base)( Prialt )
Catalog No. M24955 CAS No. 914451-03-8
Ziconotide is an analgesic agent and has been used to treat neuropathic and non-neuropathic pain. Ziconotide acts by binding to N-type calcium channels situated on the terminal part of primary afferent neurons of the nociceptive pathway therefore reducing synaptic transmission with potent antinociceptive effects.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 423 | In Stock |
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| 10MG | 605 | In Stock |
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| 25MG | 907 | In Stock |
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| 50MG | 1359 | In Stock |
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| 100MG | Get Quote | In Stock |
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| 200MG | Get Quote | In Stock |
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| 500MG | Get Quote | In Stock |
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| 1G | Get Quote | In Stock |
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Biological Information
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Product NameZiconotide Acetate (107452-89-1 free base)
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NoteResearch use only, not for human use.
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Brief DescriptionZiconotide is an analgesic agent and has been used to treat neuropathic and non-neuropathic pain. Ziconotide acts by binding to N-type calcium channels situated on the terminal part of primary afferent neurons of the nociceptive pathway therefore reducing synaptic transmission with potent antinociceptive effects.
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DescriptionZiconotide is an analgesic agent and has been used to treat neuropathic and non-neuropathic pain. Ziconotide acts by binding to N-type calcium channels situated on the terminal part of primary afferent neurons of the nociceptive pathway therefore reducing synaptic transmission with potent antinociceptive effects.
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In Vitro——
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In Vivo——
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SynonymsPrialt
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PathwayGPCR/G Protein
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TargetCalcium Channel
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RecptorN-type calcium
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Research Area——
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Indication——
Chemical Information
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CAS Number914451-03-8
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Formula Weight2639.2
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Molecular FormulaC102H172N36O32S7
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Purity>98% (HPLC)
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Solubility——
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SMILESCC1C(=O)NC(C(=O)NC2CSSCC3C(=O)NC(C(=O)NC(C(=O)NCC(=O)NC(C(=O)NC(CSSCC(C(=O)NC(CSSCC(C(=O)NC(C(=O)NCC(=O)NC(C(=O)NCC(=O)N1)CCCCN)CCCCN)N)C(=O)NC(C(=O)NCC(=O)NC(C(=O)N3)CO)C(C)O)NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(NC2=O)CO)CCCNC(=N)N)CC(C)C)CCSC)CC4=CC=C(C=C4)O)CC(=O)O)C(=O)N)CCCCN)CO)CCCNC(=N)N)CCCCN.CC(O)=O
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Brinzeu A, Berthiller J, Caillet JB, Staquet H, Mertens P. Ziconotide for spinal cord injury-related pain. Eur J Pain. 2019;23(9):1688-1700. doi:10.1002/ejp.1445
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