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G-1
CAS No. 881639-98-1
G-1( —— )
Catalog No. M24897 CAS No. 881639-98-1
G-1 is a nonsteroidal, high-affinity and selective GPR30 agonist (Ki: 11 nM).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 72 | In Stock |
|
| 10MG | 113 | In Stock |
|
| 25MG | 201 | In Stock |
|
| 50MG | 332 | In Stock |
|
| 100MG | 478 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameG-1
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NoteResearch use only, not for human use.
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Brief DescriptionG-1 is a nonsteroidal, high-affinity and selective GPR30 agonist (Ki: 11 nM).
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DescriptionG-1 is a nonsteroidal, high-affinity and selective GPR30 agonist (Ki: 11 nM).
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayCell Cycle/DNA Damage
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TargetGPR
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RecptorGPR30
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Research Area——
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Indication——
Chemical Information
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CAS Number881639-98-1
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Formula Weight412.28
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Molecular FormulaC21H18BrNO3
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Purity>98% (HPLC)
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SolubilityDMSO:50 mg/mL (121.28 mM; Need ultrasonic);H2O:< 0.1 mg/mL (insoluble)
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SMILESCC(=O)C1=CC2=C(C=C1)NC(C3C2C=CC3)C4=CC5=C(C=C4Br)OCO5
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Cheng Q, et al. G-1 exerts neuroprotective effects through G protein-coupled estrogen receptor 1 following spinal cord injury in mice. Biosci Rep. 2016 Aug 31;36(4). pii: e00373.
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