G-1

CAS No. 881639-98-1

G-1( —— )

Catalog No. M24897 CAS No. 881639-98-1

G-1 is a nonsteroidal, high-affinity and selective GPR30 agonist (Ki: 11 nM).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 72 In Stock
10MG 113 In Stock
25MG 201 In Stock
50MG 332 In Stock
100MG 478 In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    G-1
  • Note
    Research use only, not for human use.
  • Brief Description
    G-1 is a nonsteroidal, high-affinity and selective GPR30 agonist (Ki: 11 nM).
  • Description
    G-1 is a nonsteroidal, high-affinity and selective GPR30 agonist (Ki: 11 nM).
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Cell Cycle/DNA Damage
  • Target
    GPR
  • Recptor
    GPR30
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    881639-98-1
  • Formula Weight
    412.28
  • Molecular Formula
    C21H18BrNO3
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:50 mg/mL (121.28 mM; Need ultrasonic);H2O:< 0.1 mg/mL (insoluble)
  • SMILES
    CC(=O)C1=CC2=C(C=C1)NC(C3C2C=CC3)C4=CC5=C(C=C4Br)OCO5
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Cheng Q, et al. G-1 exerts neuroprotective effects through G protein-coupled estrogen receptor 1 following spinal cord injury in mice. Biosci Rep. 2016 Aug 31;36(4). pii: e00373.
molnova catalog
related products
  • PFK-158

    PFK-158 is an effective and specific inhibitor PFKFB3.

  • cangrelor tetrasodiu...

    Cangrelor tetrasodium is a reversible and selective antagonist of platelet P2Y12, with prompt and potent antiplatelet effects.cangrelor, a non-sepesific GPR17 antagonist, alleviates pulmonary fibrosis partly by inhibiting macrophage inflammation in mice.

  • Monomethyl fumarate

    Monomethyl fumarate is a potent agonist of GPR109A .