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Ritanserin
CAS No. 87051-43-2
Ritanserin( R 55667 )
Catalog No. M24881 CAS No. 87051-43-2
Ritanserin is a highly effective, relatively selective, long-acting antagonist of 5-HT2 receptor (IC50: 0.9 nM), less active on Histamine H1, Dopamine D2, Adrenergic α1, Adrenergic α2 receptors.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 49 | In Stock |
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| 2MG | 29 | In Stock |
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| 5MG | 46 | In Stock |
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| 10MG | 73 | In Stock |
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| 25MG | 147 | In Stock |
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| 50MG | 229 | In Stock |
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| 100MG | 367 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameRitanserin
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NoteResearch use only, not for human use.
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Brief DescriptionRitanserin is a highly effective, relatively selective, long-acting antagonist of 5-HT2 receptor (IC50: 0.9 nM), less active on Histamine H1, Dopamine D2, Adrenergic α1, Adrenergic α2 receptors.
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DescriptionRitanserin is a highly effective, relatively selective, long-acting antagonist of 5-HT2 receptor (IC50: 0.9 nM), less active on Histamine H1, Dopamine D2, Adrenergic α1, Adrenergic α2 receptors.
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In Vitro——
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In Vivo——
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SynonymsR 55667
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PathwayEndocrinology/Hormones
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Target5-HT Receptor
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Recptor5-HT2|D2|H1 receptor|α1-adrenergic receptor|α2 receptor
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Research Area——
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Indication——
Chemical Information
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CAS Number87051-43-2
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Formula Weight477.57
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Molecular FormulaC27H25F2N3OS
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Purity>98% (HPLC)
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SolubilityDMSO:25 mg/mL (52.35 mM; Need ultrasonic)
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SMILESCC1=C(C(N(C=CS2)C2=N1)=O)CCN(CC/3)CCC3=C(C4=CC=C(F)C=C4)\C5=CC=C(F)C=C5
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Leysen JE, et al. Receptor-binding properties in vitro and in vivo of ritanserin: A very potent and long acting serotonin-S2 antagonist. Mol Pharmacol. 1985 Jun;27(6):600-11.
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