TPPB

CAS No. 497259-23-1

TPPB( —— )

Catalog No. M24458 CAS No. 497259-23-1

TPPB is a kinase C activator of cell-permeable benzolactam-derived protein (Ki: 11.9 nM).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 560 In Stock
5MG 519 In Stock
10MG 748 In Stock
100MG Get Quote In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    TPPB
  • Note
    Research use only, not for human use.
  • Brief Description
    TPPB is a kinase C activator of cell-permeable benzolactam-derived protein (Ki: 11.9 nM).
  • Description
    TPPB is a kinase C activator of cell-permeable benzolactam-derived protein (Ki: 11.9 nM).
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Angiogenesis
  • Target
    PKC
  • Recptor
    PKC
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    497259-23-1
  • Formula Weight
    501.54
  • Molecular Formula
    C27H30F3N3O3
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:125 mg/mL (249.23 mM; Need ultrasonic)
  • SMILES
    CC(C)[C@@H](C(N[C@H](CO)C1)=O)N(C)c(cc2)c1cc2NC(/C=C/C=C/c1ccc(C(F)(F)F)cc1)=O
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Kozikowski AP, et al. New amide-bearing benzolactam-based protein kinase C modulators induce enhanced secretion of the amyloid precursor protein metabolite sAPPalpha. J Med Chem. 2003 Jan 30;46(3):364-73.
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