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TPPB
CAS No. 497259-23-1
TPPB( —— )
Catalog No. M24458 CAS No. 497259-23-1
TPPB is a kinase C activator of cell-permeable benzolactam-derived protein (Ki: 11.9 nM).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 560 | In Stock |
|
| 5MG | 519 | In Stock |
|
| 10MG | 748 | In Stock |
|
| 100MG | Get Quote | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameTPPB
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NoteResearch use only, not for human use.
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Brief DescriptionTPPB is a kinase C activator of cell-permeable benzolactam-derived protein (Ki: 11.9 nM).
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DescriptionTPPB is a kinase C activator of cell-permeable benzolactam-derived protein (Ki: 11.9 nM).
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayAngiogenesis
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TargetPKC
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RecptorPKC
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Research Area——
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Indication——
Chemical Information
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CAS Number497259-23-1
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Formula Weight501.54
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Molecular FormulaC27H30F3N3O3
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Purity>98% (HPLC)
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SolubilityDMSO:125 mg/mL (249.23 mM; Need ultrasonic)
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SMILESCC(C)[C@@H](C(N[C@H](CO)C1)=O)N(C)c(cc2)c1cc2NC(/C=C/C=C/c1ccc(C(F)(F)F)cc1)=O
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Kozikowski AP, et al. New amide-bearing benzolactam-based protein kinase C modulators induce enhanced secretion of the amyloid precursor protein metabolite sAPPalpha. J Med Chem. 2003 Jan 30;46(3):364-73.
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