TRPM4-IN-1( CBA | 4-chloro-2-(2-(2-chlorophenoxy)acetamido)benzoic acid )

Catalog No. M24301 CAS No. 351424-20-9

TRPM4-IN-1 is a potent and selective inhibitor of TRPM4 with an IC50 of 1.5 μM.

Purity : >98% (HPLC)

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

Size	Price / USD	Stock	Quantity
1 mL x 10 mM in DMSO	64	In Stock
5MG	36	In Stock
10MG	58	In Stock
25MG	126	In Stock
50MG	210	In Stock
100MG	338	In Stock
200MG	492	In Stock
500MG	Get Quote	In Stock
1G	Get Quote	In Stock

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Biological Information

Product Name

TRPM4-IN-1
Note

Research use only, not for human use.
Brief Description

TRPM4-IN-1 is a potent and selective inhibitor of TRPM4 with an IC50 of 1.5 μM.
Description

TRPM4-IN-1 is a potent and selective inhibitor of TRPM4 with an IC50 of 1.5 μM.
In Vitro

Western Blot Analysis Cell Line:HEK293 cells Concentration:50 μM Incubation Time:Overnight Result:Partial rescued the total and surface expression of A432T.
In Vivo

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Synonyms

CBA | 4-chloro-2-(2-(2-chlorophenoxy)acetamido)benzoic acid
Pathway

Membrane Transporter/Ion Channel
Target

TRP/TRPV Channel
Recptor

TRPM4
Research Area

——
Indication

——

Chemical Information

CAS Number

351424-20-9
Formula Weight

340.16
Molecular Formula

C15H11Cl2NO4
Purity

>98% (HPLC)
Solubility

DMSO:80mg/ml(235.18mM; need ultrasonic)
SMILES

OC(c(ccc(Cl)c1)c1NC(COc(cccc1)c1Cl)=O)=O
Chemical Name

——

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

1.Ozhathil L C , Delalande C , Bianchi B , et al. Identification of potent and selective small molecule inhibitors of the cation channel TRPM4[J]. British Journal of Pharmacology, 2018.

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