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TRPM4-IN-1

CAS No. 351424-20-9

TRPM4-IN-1( CBA | 4-chloro-2-(2-(2-chlorophenoxy)acetamido)benzoic acid )

Catalog No. M24301 CAS No. 351424-20-9

TRPM4-IN-1 is a potent and selective inhibitor of TRPM4 with an IC50 of 1.5 μM.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 64 In Stock
5MG 36 In Stock
10MG 58 In Stock
25MG 126 In Stock
50MG 210 In Stock
100MG 338 In Stock
200MG 492 In Stock
500MG Get Quote In Stock
1G Get Quote In Stock
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Biological Information

  • Product Name
    TRPM4-IN-1
  • Note
    Research use only, not for human use.
  • Brief Description
    TRPM4-IN-1 is a potent and selective inhibitor of TRPM4 with an IC50 of 1.5 μM.
  • Description
    TRPM4-IN-1 is a potent and selective inhibitor of TRPM4 with an IC50 of 1.5 μM.
  • In Vitro
    Western Blot Analysis Cell Line:HEK293 cells Concentration:50 μM Incubation Time:Overnight Result:Partial rescued the total and surface expression of A432T.
  • In Vivo
    ——
  • Synonyms
    CBA | 4-chloro-2-(2-(2-chlorophenoxy)acetamido)benzoic acid
  • Pathway
    Membrane Transporter/Ion Channel
  • Target
    TRP/TRPV Channel
  • Recptor
    TRPM4
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    351424-20-9
  • Formula Weight
    340.16
  • Molecular Formula
    C15H11Cl2NO4
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:80mg/ml(235.18mM; need ultrasonic)
  • SMILES
    OC(c(ccc(Cl)c1)c1NC(COc(cccc1)c1Cl)=O)=O
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Ozhathil L C , Delalande C , Bianchi B , et al. Identification of potent and selective small molecule inhibitors of the cation channel TRPM4[J]. British Journal of Pharmacology, 2018.
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