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TRPM4-IN-1
CAS No. 351424-20-9
TRPM4-IN-1( CBA | 4-chloro-2-(2-(2-chlorophenoxy)acetamido)benzoic acid )
Catalog No. M24301 CAS No. 351424-20-9
TRPM4-IN-1 is a potent and selective inhibitor of TRPM4 with an IC50 of 1.5 μM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 34 | In Stock |
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| 10MG | 55 | In Stock |
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| 25MG | 120 | In Stock |
|
| 50MG | 203 | In Stock |
|
| 100MG | 327 | In Stock |
|
| 200MG | 476 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameTRPM4-IN-1
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NoteResearch use only, not for human use.
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Brief DescriptionTRPM4-IN-1 is a potent and selective inhibitor of TRPM4 with an IC50 of 1.5 μM.
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DescriptionTRPM4-IN-1 is a potent and selective inhibitor of TRPM4 with an IC50 of 1.5 μM.
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In VitroWestern Blot Analysis Cell Line:HEK293 cells Concentration:50 μM Incubation Time:Overnight Result:Partial rescued the total and surface expression of A432T.
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In Vivo——
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SynonymsCBA | 4-chloro-2-(2-(2-chlorophenoxy)acetamido)benzoic acid
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PathwayMembrane Transporter/Ion Channel
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TargetTRP/TRPV Channel
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RecptorTRPM4
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Research Area——
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Indication——
Chemical Information
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CAS Number351424-20-9
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Formula Weight340.16
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Molecular FormulaC15H11Cl2NO4
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Purity>98% (HPLC)
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SolubilityDMSO:80mg/ml(235.18mM; need ultrasonic)
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SMILESOC(c(ccc(Cl)c1)c1NC(COc(cccc1)c1Cl)=O)=O
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Ozhathil L C , Delalande C , Bianchi B , et al. Identification of potent and selective small molecule inhibitors of the cation channel TRPM4[J]. British Journal of Pharmacology, 2018.
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