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Pimethixene

CAS No. 314-03-4

Pimethixene( Pimetixene | Calmixen )

Catalog No. M24244 CAS No. 314-03-4

Pimethixene is a highly potent 5-HT1A, 5-HT2A, 5-HT2B, 5-HT2C, histamine H1, dopamine D2 and D4.4 as well as muscarinic M1 and M2 receptors antagonist(pKis of 7.63, 10.22, 10.44, 8.42, 10.14, 8.19, 7.54, 8.61 and 9.38, respectively).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 46 In Stock
2MG 28 In Stock
5MG 41 In Stock
10MG 56 In Stock
25MG 103 In Stock
50MG 149 In Stock
100MG 221 In Stock
200MG 331 In Stock
500MG Get Quote In Stock
1G Get Quote In Stock
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Biological Information

  • Product Name
    Pimethixene
  • Note
    Research use only, not for human use.
  • Brief Description
    Pimethixene is a highly potent 5-HT1A, 5-HT2A, 5-HT2B, 5-HT2C, histamine H1, dopamine D2 and D4.4 as well as muscarinic M1 and M2 receptors antagonist(pKis of 7.63, 10.22, 10.44, 8.42, 10.14, 8.19, 7.54, 8.61 and 9.38, respectively).
  • Description
    Pimethixene is a highly potent 5-HT1A, 5-HT2A, 5-HT2B, 5-HT2C, histamine H1, dopamine D2 and D4.4 as well as muscarinic M1 and M2 receptors antagonist(pKis of 7.63, 10.22, 10.44, 8.42, 10.14, 8.19, 7.54, 8.61 and 9.38, respectively).
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    Pimetixene | Calmixen
  • Pathway
    Endocrinology/Hormones
  • Target
    5-HT Receptor
  • Recptor
    5-HT2A Receptor|5-HT2B Receptor|5-HT2C Receptor|H1 receptor|5-HT1A Receptor|D2 receptor|DD4.4 receptor|M1 receptor|M2 receptor
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    314-03-4
  • Formula Weight
    293.43
  • Molecular Formula
    C19H19NS
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    CN(CC1)CCC1=C1c(cccc2)c2Sc2c1cccc2
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Schmitz B, et al. BF-1--a novel selective 5-HT2B receptor antagonist blocking neurogenic dural plasma protein extravasation in guinea pigs. Eur J Pharmacol. 2015 Mar 15;751:73-80.
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