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Pericyazine
CAS No. 2622-26-6
Pericyazine( Propericiazine | RP 8909 )
Catalog No. M24171 CAS No. 2622-26-6
Pericyazine is a selective D2-dopamine receptor antagonist. Pericyazine is a first-generation antipsychotic drug that is used as an adjunct to the short-term management of severe anxiety states and psychosis.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 67 | In Stock |
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| 2MG | 51 | In Stock |
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| 5MG | 81 | In Stock |
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| 10MG | 120 | In Stock |
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| 25MG | 235 | In Stock |
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| 50MG | 380 | In Stock |
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| 100MG | 554 | In Stock |
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| 200MG | Get Quote | In Stock |
|
| 500MG | 1200 | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NamePericyazine
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NoteResearch use only, not for human use.
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Brief DescriptionPericyazine is a selective D2-dopamine receptor antagonist. Pericyazine is a first-generation antipsychotic drug that is used as an adjunct to the short-term management of severe anxiety states and psychosis.
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DescriptionPericyazine is a selective D2-dopamine receptor antagonist. Pericyazine is a first-generation antipsychotic drug that is used as an adjunct to the short-term management of severe anxiety states and psychosis.
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In Vitro——
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In VivoStudies in rodents show that Pericyazine is able to produce potentiation of ether and hexobarbital narcosis and morphine analgesia. It also has hypothermic activity and produces depression of spontaneous motor activity in mice. On a milligram potency basis, Pericyazine is more potent than chlorpromizine in the potentiation of barbiturate narcosis test and the blocking of conditioned avoidance in rats. Pericyazine demonstrates analgesic properties similar to methotrimeprazine in mice and rats and produces adrenergic blocking effects in mice and dogs.
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SynonymsPropericiazine | RP 8909
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PathwayGPCR/G Protein
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TargetDopamine Receptor
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RecptorD2-dopamine receptor
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Research Area——
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Indication——
Chemical Information
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CAS Number2622-26-6
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Formula Weight365.49
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Molecular FormulaC21H23N3OS
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Purity>98% (HPLC)
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SolubilityDMSO:200 mg/mL (547.21 mM; Need ultrasonic)
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SMILESN#Cc(cc1)cc2c1Sc(cccc1)c1N2CCCN(CC1)CCC1O
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Morley KC, et al. Pericyazine in the treatment of cannabis dependence in general practice: a naturalistic pilot trial. Subst Abuse Rehabil. 2012 May 28;3:43-7.
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