Pericyazine

CAS No. 2622-26-6

Pericyazine( Propericiazine | RP 8909 )

Catalog No. M24171 CAS No. 2622-26-6

Pericyazine is a selective D2-dopamine receptor antagonist. Pericyazine is a first-generation antipsychotic drug that is used as an adjunct to the short-term management of severe anxiety states and psychosis.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 67 In Stock
2MG 51 In Stock
5MG 81 In Stock
10MG 120 In Stock
25MG 235 In Stock
50MG 380 In Stock
100MG 554 In Stock
200MG Get Quote In Stock
500MG 1200 In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    Pericyazine
  • Note
    Research use only, not for human use.
  • Brief Description
    Pericyazine is a selective D2-dopamine receptor antagonist. Pericyazine is a first-generation antipsychotic drug that is used as an adjunct to the short-term management of severe anxiety states and psychosis.
  • Description
    Pericyazine is a selective D2-dopamine receptor antagonist. Pericyazine is a first-generation antipsychotic drug that is used as an adjunct to the short-term management of severe anxiety states and psychosis.
  • In Vitro
    ——
  • In Vivo
    Studies in rodents show that Pericyazine is able to produce potentiation of ether and hexobarbital narcosis and morphine analgesia. It also has hypothermic activity and produces depression of spontaneous motor activity in mice. On a milligram potency basis, Pericyazine is more potent than chlorpromizine in the potentiation of barbiturate narcosis test and the blocking of conditioned avoidance in rats. Pericyazine demonstrates analgesic properties similar to methotrimeprazine in mice and rats and produces adrenergic blocking effects in mice and dogs.
  • Synonyms
    Propericiazine | RP 8909
  • Pathway
    GPCR/G Protein
  • Target
    Dopamine Receptor
  • Recptor
    D2-dopamine receptor
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    2622-26-6
  • Formula Weight
    365.49
  • Molecular Formula
    C21H23N3OS
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:200 mg/mL (547.21 mM; Need ultrasonic)
  • SMILES
    N#Cc(cc1)cc2c1Sc(cccc1)c1N2CCCN(CC1)CCC1O
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Morley KC, et al. Pericyazine in the treatment of cannabis dependence in general practice: a naturalistic pilot trial. Subst Abuse Rehabil. 2012 May 28;3:43-7.
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