PF-06882961 Tris

CAS No. 2230198-03-3

PF-06882961 Tris( UNII-2HJV78O0SS )

Catalog No. M24014 CAS No. 2230198-03-3

PF-06882961 Tris is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 287 In Stock
10MG 430 In Stock
25MG 710 In Stock
50MG 977 In Stock
100MG 1321 In Stock
200MG Get Quote In Stock
500MG 2632 In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    PF-06882961 Tris
  • Note
    Research use only, not for human use.
  • Brief Description
    PF-06882961 Tris is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.
  • Description
    PF-06882961 Tris is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    UNII-2HJV78O0SS
  • Pathway
    GPCR/G Protein
  • Target
    Glucagon Receptor
  • Recptor
    GLP-1
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    2230198-03-3
  • Formula Weight
    676.7
  • Molecular Formula
    C35H41FN6O7
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:10 mM
  • SMILES
    C1CO[C@@H]1CN2C3=C(C=CC(=C3)C(=O)O)N=C2CN4CCC(CC4)C5=NC(=CC=C5)OCC6=C(C=C(C=C6)C#N)F.C(C(CO)(CO)N)O
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Méndez M, Matter H, Defossa E, et al. Design, Synthesis, and Pharmacological Evaluation of Potent Positive Allosteric Modulators of the Glucagon-like Peptide-1 Receptor (GLP-1R). J Med Chem. 2020;63(5):2292-2307. doi:10.1021/acs.jmedchem.9b01071
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