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Desketoraloxifene
CAS No. 216570-81-9
Desketoraloxifene( —— )
Catalog No. M23980 CAS No. 216570-81-9
Desketoraloxifene is a selective estrogen receptor modulator, inhibiting mammalian PLD (PLD1 and PLD2).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 272 | In Stock |
|
| 10MG | 409 | In Stock |
|
| 25MG | 737 | In Stock |
|
| 100MG | Get Quote | In Stock |
|
| 200MG | Get Quote | In Stock |
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| 500MG | Get Quote | In Stock |
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| 1G | Get Quote | In Stock |
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Biological Information
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Product NameDesketoraloxifene
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NoteResearch use only, not for human use.
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Brief DescriptionDesketoraloxifene is a selective estrogen receptor modulator, inhibiting mammalian PLD (PLD1 and PLD2).
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DescriptionDesketoraloxifene is a selective estrogen receptor modulator, inhibiting mammalian PLD (PLD1 and PLD2).
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayMetabolic Enzyme/Protease
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TargetPhospholipase
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RecptorPLD1|PLD2
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Research Area——
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Indication——
Chemical Information
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CAS Number216570-81-9
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Formula Weight445.57
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Molecular FormulaC27H27NO3S
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Purity>98% (HPLC)
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Solubility——
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SMILESC1CCN(CC1)CCOC2=CC=C(C=C2)C3=C(SC4=C3C=CC(=C4)O)C5=CC=C(C=C5)O
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Scott S A , Spencer C T , MC O’Reilly, et al. Discovery of Desketoraloxifene Analogues as Inhibitorsof Mammalian, Pseudomonas aeruginosa, and NAPE PhospholipaseD Enzymes[J]. Acs Chemical Biology, 2015, 10(2):421.
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