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LSD1-IN-7 benzenesulfonate
CAS No. 2097523-60-7
LSD1-IN-7 benzenesulfonate( CC-90011 benzenesulfonate )
Catalog No. M23947 CAS No. 2097523-60-7
LSD1-IN-7 benzenesulfonate is a potent and orally active inhibitor of lysine specific demethylase-1 (LSD1) with anticancer activity.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 170 | In Stock |
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| 2MG | 74 | In Stock |
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| 5MG | 120 | In Stock |
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| 10MG | 188 | In Stock |
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| 25MG | 330 | In Stock |
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| 50MG | 479 | In Stock |
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| 100MG | 695 | In Stock |
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| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameLSD1-IN-7 benzenesulfonate
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NoteResearch use only, not for human use.
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Brief DescriptionLSD1-IN-7 benzenesulfonate is a potent and orally active inhibitor of lysine specific demethylase-1 (LSD1) with anticancer activity.
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DescriptionLSD1-IN-7 benzenesulfonate is a potent and orally active inhibitor of lysine specific demethylase-1 (LSD1) with anticancer activity.
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In Vitro——
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In VivoAnimal Model:BALB/c nude mice bearing small cell lung carcinoma (SCLC)Dosage:5 mg/kg Administration:Oral administration; daily; for 30 days Result:Showed a tumor growth inhibition (TGI) of 78% at 5 mg/kg with nobody weight loss.
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SynonymsCC-90011 benzenesulfonate
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PathwayChromatin/Epigenetic
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TargetHistone Demethylase
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RecptorLSD1
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Research Area——
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Indication——
Chemical Information
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CAS Number2097523-60-7
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Formula Weight609.64
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Molecular FormulaC30H29F2N5O5S
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Purity>98% (HPLC)
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SolubilityDMSO:60mg/ml(98.42mM; Need ultrasonic)
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SMILESN#CC1=CC=C(C(N=C(N2CCC(N)CC2)N3C)=C(C4=CC=C(OC)C(F)=C4)C3=O)C=C1F.O=S(C5=CC=CC=C5)(O)=O
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Young K. Chen, et al. Compositions comprising an inhibitor of lysine specific demethylase-1. WO2017079670A1.
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