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KAN0438757
CAS No. 1451255-59-6
KAN0438757( —— )
Catalog No. M23618 CAS No. 1451255-59-6
KAN0438757 is a selective and potent inhibitor of the metabolic kinase PFKFB3 with an IC50 of 0.19 μM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 206 | In Stock |
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| 5MG | 192 | In Stock |
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| 10MG | 307 | In Stock |
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| 25MG | 554 | In Stock |
|
| 50MG | 745 | In Stock |
|
| 100MG | 1014 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameKAN0438757
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NoteResearch use only, not for human use.
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Brief DescriptionKAN0438757 is a selective and potent inhibitor of the metabolic kinase PFKFB3 with an IC50 of 0.19 μM.
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DescriptionKAN0438757 is a selective and potent inhibitor of the metabolic kinase PFKFB3 with an IC50 of 0.19 μM.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayCytoskeleton/Cell Adhesion Molecules
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TargetGlucokinase
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RecptorPFKFB3
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Research Area——
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Indication——
Chemical Information
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CAS Number1451255-59-6
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Formula Weight447.43
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Molecular FormulaC21H18FNO7S
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Purity>98% (HPLC)
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SolubilityDMSO:130 mg/mL (290.55 mM; Need ultrasonic)
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SMILESC1=CC(=CC(=C1)S(=O)(=O)NC2=CC(=C(C=C2)C(=O)OCCO)O)C3=C(C=CC(=C3)F)O
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Gustafsson NMS, et al. Targeting PFKFB3 radiosensitizes cancer cells and suppresses homologous recombination. Nat Commun. 2018 Sep 24;9(1):3872.
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