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Home - Products - Metabolic Enzyme/Protease - Dehydrogenase - AG-120 (racemic)

AG-120 (racemic)

CAS No. 1448346-63-1

AG-120 (racemic)( —— )

Catalog No. M23614 CAS No. 1448346-63-1

AG-120 (racemic), the racemic mixture of AG-120, is an orally available isocitrate dehydrogenase type 1 (IDH1) inhibitor, and shows potential antineoplastic activity.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 93 In Stock
5MG 69 In Stock
10MG 107 In Stock
25MG 180 In Stock
50MG 263 In Stock
100MG 390 In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G Get Quote In Stock
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Biological Information

  • Product Name
    AG-120 (racemic)
  • Note
    Research use only, not for human use.
  • Brief Description
    AG-120 (racemic), the racemic mixture of AG-120, is an orally available isocitrate dehydrogenase type 1 (IDH1) inhibitor, and shows potential antineoplastic activity.
  • Description
    AG-120 (racemic), the racemic mixture of AG-120, is an orally available isocitrate dehydrogenase type 1 (IDH1) inhibitor, and shows potential antineoplastic activity.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Metabolic Enzyme/Protease
  • Target
    Dehydrogenase
  • Recptor
    IDH1
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1448346-63-1
  • Formula Weight
    582.96
  • Molecular Formula
    C28H22ClF3N6O3
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:100 mg/ml (171.54 mM); Ethanol:100 mg/ml (171.54 mM)
  • SMILES
    O=C1CC[C@@H](C(N(C(C(NC2CC(F)(F)C2)=O)C3=CC=CC=C3Cl)C4=CC(F)=CN=C4)=O)N1C5=NC=CC(C#N)=C5
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.M Cecilia Caino, Dario C Altieri. Clin Cancer Res. 2016 Feb 1;22(3):540-5.
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