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CIM0216
CAS No. 1031496-06-6
CIM0216( N-(5-methyl-1,2-oxazol-3-yl)-2-phenyl-2-(1,2,3,4-tetrahydroquinolin-1-yl)acetamide )
Catalog No. M23235 CAS No. 1031496-06-6
CIM0216 is a synthetic TRPM3 activator whose potency and apparent affinity greatly exceeds that of the canonical TRPM3 agonist.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 88 | In Stock |
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| 2MG | 51 | In Stock |
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| 5MG | 80 | In Stock |
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| 10MG | 141 | In Stock |
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| 25MG | 297 | In Stock |
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| 50MG | 456 | In Stock |
|
| 100MG | 686 | In Stock |
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| 200MG | Get Quote | In Stock |
|
| 500MG | 1423 | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameCIM0216
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NoteResearch use only, not for human use.
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Brief DescriptionCIM0216 is a synthetic TRPM3 activator whose potency and apparent affinity greatly exceeds that of the canonical TRPM3 agonist.
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DescriptionCIM0216 is a synthetic TRPM3 activator whose potency and apparent affinity greatly exceeds that of the canonical TRPM3 agonist.
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In Vitro——
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In Vivo——
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SynonymsN-(5-methyl-1,2-oxazol-3-yl)-2-phenyl-2-(1,2,3,4-tetrahydroquinolin-1-yl)acetamide
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PathwayMembrane Transporter/Ion Channel
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TargetTRP/TRPV Channel
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RecptorTRPM3
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Research Area——
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Indication——
Chemical Information
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CAS Number1031496-06-6
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Formula Weight347.41
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Molecular FormulaC21H21N3O2
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Purity>98% (HPLC)
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SolubilityDMSO: 30 mg/mL?(86.35 mM;?Need ultrasonic and warming);Ethanol: 17 mg/mL?(48.93 mM;?Need ultrasonic and warming)
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SMILESO=C(NC1=NOC(C)=C1)C(C2=CC=CC=C2)N3CCCC4=C3C=CC=C4
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Vriens J , Owsianik G , Hofmann T , et al. TRPM3 is a nociceptor channel involved in the detection of noxious heat.[J]. Neuron, 2011, 70(3):482-494.
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