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Taltirelin acetate
CAS No. 1549593-23-8
Taltirelin acetate( TA-0910 acetate )
Catalog No. M22365 CAS No. 1549593-23-8
Taltirelin acetate is a superagonist at thyrotropin-releasing hormone receptor (TRH-R)(IC50 of 910 nM and EC50 of 36 nM for stimulating an increase in cytosolic Ca2+ concentration (Ca2+ release)).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 49 | In Stock |
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| 2MG | 29 | In Stock |
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| 5MG | 45 | In Stock |
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| 10MG | 73 | In Stock |
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| 25MG | 144 | In Stock |
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| 50MG | 237 | In Stock |
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| 100MG | 369 | In Stock |
|
| 200MG | 547 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameTaltirelin acetate
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NoteResearch use only, not for human use.
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Brief DescriptionTaltirelin acetate is a superagonist at thyrotropin-releasing hormone receptor (TRH-R)(IC50 of 910 nM and EC50 of 36 nM for stimulating an increase in cytosolic Ca2+ concentration (Ca2+ release)).
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DescriptionTaltirelin acetate is a superagonist at thyrotropin-releasing hormone receptor (TRH-R)(IC50 of 910 nM and EC50 of 36 nM for stimulating an increase in cytosolic Ca2+ concentration (Ca2+ release)).
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In Vitro——
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In Vivo——
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SynonymsTA-0910 acetate
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PathwayOthers
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TargetOther Targets
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RecptorTHR
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Research AreaNervous system
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IndicationSpinocerebellar Degeneration
Chemical Information
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CAS Number1549593-23-8
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Formula Weight465.46
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Molecular FormulaC19H27N7O7
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Purity>98% (HPLC)
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SolubilityDMSO:125 mg/mL (268.55 mM; Need ultrasonic)
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SMILESO=C(N(CCC1)[C@@H]1C(N)=O)[C@@H](NC([C@@H](NC2=O)CC(N2C)=O)=O)CC3=CN=CN3.CC(O)=O
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Thirunarayanan N, et al. Taltirelin is a superagonist at the human thyrotropin-releasing hormone receptor. Front Endocrinol (Lausanne). 2012 Oct 9;3:120.
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