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Spastazoline
CAS No. 2351882-11-4
Spastazoline( —— )
Catalog No. M21959 CAS No. 2351882-11-4
Spastazoline is a potent and selective inhibitor of spastin(Human spastin with IC50 of 99 nM ).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 71 | In Stock |
|
| 5MG | 65 | In Stock |
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| 10MG | 107 | In Stock |
|
| 25MG | 216 | In Stock |
|
| 50MG | 317 | In Stock |
|
| 100MG | 455 | In Stock |
|
| 200MG | 631 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameSpastazoline
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NoteResearch use only, not for human use.
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Brief DescriptionSpastazoline is a potent and selective inhibitor of spastin(Human spastin with IC50 of 99 nM ).
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DescriptionSpastazoline is a potent and selective inhibitor of spastin(Human spastin with IC50 of 99 nM).
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayOthers
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TargetOther Targets
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Recptorspastin
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Research Area——
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Indication——
Chemical Information
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CAS Number2351882-11-4
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Formula Weight382.51
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Molecular FormulaC20H30N8
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Purity>98% (HPLC)
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SolubilityDMSO:95 mg/ml(248.36 mM; Need ultrasonic)
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SMILESCC(C)[C@@H]1CN(CCN1)c1nc(Nc2cc([nH]n2)C(C)(C)C)c2cc[nH]c2n1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Cupido T, et al. Designing a chemical inhibitor for the AAA protein spastin using active site mutations. Nat Chem Biol. 2019 Feb 18.2. Pisa R , Cupido T , Steinman J B , et al. Analyzing Resistance to Design Selective Chemical Inhibitors for AAA Proteins[J]. Cell Chemical Biology, 2019, 26(9).
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