Cart
sales@molnova.com
H-9 hydrochloride
CAS No. 116970-50-4
H-9 hydrochloride( —— )
Catalog No. M21838 CAS No. 116970-50-4
H-9 hydrochloride inhibits PKA (Ki=1.9 μM), PKC (Ki=18 μM; cGKI (PKG) =0.87 μM; MLCK=70 μM).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 10MG | 76 | In Stock |
|
| 50MG | 320 | In Stock |
|
| 100MG | Get Quote | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
-
Product NameH-9 hydrochloride
-
NoteResearch use only, not for human use.
-
Brief DescriptionH-9 hydrochloride inhibits PKA (Ki=1.9 μM), PKC (Ki=18 μM; cGKI (PKG) =0.87 μM; MLCK=70 μM).
-
DescriptionH-9 hydrochloride inhibits PKA (Ki=1.9 μM), PKC (Ki=18 μM; cGKI (PKG) =0.87 μM; MLCK=70 μM). It has shown to dramatically reduce the GABA response of GABAA currents in retinal rod bipolar cells as well as inhibit smooth muscle cell relaxation induced by cGRP. H-9 dihydrochloride has also been used for purification of protein kinases in ligand affinity chromatography.
-
In Vitro——
-
In Vivo——
-
Synonyms——
-
PathwayOthers
-
TargetOther Targets
-
RecptorcGKI
-
Research Area——
-
Indication——
Chemical Information
-
CAS Number116970-50-4
-
Formula Weight287.77
-
Molecular FormulaC11H13N3O2S?HCl
-
Purity>98% (HPLC)
-
Solubility——
-
SMILESC1=CC2=C(C=CN=C2)C(=C1)S(=O)(=O)NCCN.Cl
-
Chemical Name——
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
1. Wolf, M., et al. 1985. J. Biol. Chem. 260: 15718-15722. PMID: 4066694
2. Inagaki, M., et al. 1985. J. Biol. Chem. 260: 2922-2925. PMID: 2982842
3. Gillette, M.A., et al. 1996. J. Neurophysiol. 76: 3070-3086. PMID: 8930256
molnova catalog
related products
-
Terrestriamide
Terrestriamide
-
RR-11a analog
RR-11a analog is a potent and selective asparaginyl endopeptidases (AE) (Legumain) inhibitors(IC50 values of 4.5 nM, 4.5 nM and 31 nM for AE1 in Trichomonas Vaginalis, AE in Ixodes ricinus and AE in Schistosoma mansoni, respectively).
-
R-G-D-T
R-G-D-T
