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Home - Products - Cell Cycle/DNA Damage - Potassium Channel - A2764 dihydrochloride

A2764 dihydrochloride

CAS No. 861038-72-4

A2764 dihydrochloride( —— )

Catalog No. M21057 CAS No. 861038-72-4

A2764 dihydrochloride is a highly selective inhibitor of TRESK.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 37 In Stock
5MG 33 In Stock
10MG 55 In Stock
25MG 98 In Stock
50MG 161 In Stock
100MG 250 In Stock
200MG 358 In Stock
500MG Get Quote In Stock
1G Get Quote In Stock
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Biological Information

  • Product Name
    A2764 dihydrochloride
  • Note
    Research use only, not for human use.
  • Brief Description
    A2764 dihydrochloride is a highly selective inhibitor of TRESK.
  • Description
    A2764 dihydrochloride is a highly selective inhibitor of TRESK.
  • In Vitro
    A2764 (100 μM) inhibits the background K+ current by 42.8±11.5% when it applies to the oocytes expressing mTRESK.A2764 (100 μM) shows an improvedinhibitory potency for activated channel with an IC50 of activated channel in ionomycin-activated mTRESK current.The subsequent application of A2764 strongly inhibits the current (77.8±3.5%).A2764 (100 μM) inhibits the current of TRESK under resting conditions and in the activated state by 42.8±11.5% and 77.8±3.5%, respectively.
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Cell Cycle/DNA Damage
  • Target
    Potassium Channel
  • Recptor
    mTRESK channel
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    861038-72-4
  • Formula Weight
    351.7
  • Molecular Formula
    C15H21Cl3N2O
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:41.67 mg/mL?(118.48 mM)
  • SMILES
    CCN(CC)CCOc1ccc(Cl)c2cccnc12.Cl.Cl
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Chemically Modified Derivatives of the Activator Compound Cloxyquin Exert Inhibitory Effect on TRESK (K2P18.1) Background Potassium Channel.[J]. Molecular pharmacology 2019.
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