R1487

CAS No. 449811-92-1

R1487( —— )

Catalog No. M20961 CAS No. 449811-92-1

R1487 is an orally bioavailable and highly selective p38α mitogen-activated protein kinase inhibitor.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 283 In Stock
10MG 430 In Stock
25MG 710 In Stock
50MG 977 In Stock
100MG 1321 In Stock
200MG Get Quote In Stock
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Biological Information

  • Product Name
    R1487
  • Note
    Research use only, not for human use.
  • Brief Description
    R1487 is an orally bioavailable and highly selective p38α mitogen-activated protein kinase inhibitor.
  • Description
    R1487 is an orally bioavailable and highly selective p38α mitogen-activated protein kinase inhibitor.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    MAPK/ERK Signaling
  • Target
    p38 MAPK
  • Recptor
    p38α
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    449811-92-1
  • Formula Weight
    388.36
  • Molecular Formula
    C19H18F2N4O3
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    Cn1c(=O)c(Oc2ccc(F)cc2F)cc2cnc(NC3CCOCC3)nc21
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Dunford E C Herbst E A Jeoung N H et al. PDH activation during in vitro muscle contractions in PDH kinase 2 knockout mice: Effect of PDH kinase 1 compensation[J]. American Journal of Physiology Regulatory Integrative & Comparative Physiology 2011 300(6):R1487.
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